日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Acetylation reprograms MITF target selectivity and residence time

乙酰化作用会改变MITF靶标选择性和停留时间。

Pakavarin Louphrasitthiphol ,Alessia Loffreda ,Vivian Pogenberg ,Sarah Picaud ,Alexander Schepsky ,Hans Friedrichsen ,Zhiqiang Zeng ,Anahita Lashgari ,Benjamin Thomas ,E Elizabeth Patton ,Matthias Wilmanns ,Panagis Filippakopoulos ,Jean-Philippe Lambert ,Eiríkur Steingrímsson ,Davide Mazza ,Colin R Goding

Aminopeptidase Expression in Multiple Myeloma Associates with Disease Progression and Sensitivity to Melflufen

多发性骨髓瘤中的氨基肽酶表达与疾病进展和对美氟芬的敏感性相关

Juho J Miettinen, Romika Kumari, Gunnhildur Asta Traustadottir, Maiju-Emilia Huppunen, Philipp Sergeev, Muntasir M Majumder, Alexander Schepsky, Thorarinn Gudjonsson, Juha Lievonen, Despina Bazou, Paul Dowling, Peter O Gorman, Ana Slipicevic, Pekka Anttila, Raija Silvennoinen, Nina N Nupponen, Fredr

Tuning Transcription Factor Availability through Acetylation-Mediated Genomic Redistribution

通过乙酰化介导的基因组重分布来调节转录因子可用性

Pakavarin Louphrasitthiphol ,Robert Siddaway ,Alessia Loffreda ,Vivian Pogenberg ,Hans Friedrichsen ,Alexander Schepsky ,Zhiqiang Zeng ,Min Lu ,Thomas Strub ,Rasmus Freter ,Richard Lisle ,Eda Suer ,Benjamin Thomas ,Benjamin Schuster-Böckler ,Panagis Filippakopoulos ,Mark Middleton ,Xin Lu ,E Elizabeth Patton ,Irwin Davidson ,Jean-Philippe Lambert ,Matthias Wilmanns ,Eiríkur Steingrímsson ,Davide Mazza ,Colin R Goding

Melflufen, a peptide-conjugated alkylator, is an efficient anti-neo-plastic drug in breast cancer cell lines

Melflufen 是一种肽结合烷基化剂,是乳腺癌细胞系中有效的抗肿瘤药物

Alexander Schepsky, Gunnhildur Asta Traustadottir, Jon Petur Joelsson, Saevar Ingthorsson, Jennifer Kricker, Jon Thor Bergthorsson, Arni Asbjarnarson, Thorkell Gudjonsson, Nina Nupponen, Ana Slipicevic, Fredrik Lehmann, Thorarinn Gudjonsson

Subcellular localization and stability of MITF are modulated by the bHLH-Zip domain

MITF 的亚细胞定位和稳定性受 bHLH-Zip 结构域调节

Valerie Fock, Sigurdur Runar Gudmundsson, Hilmar Orn Gunnlaugsson, Jon August Stefansson, Vivien Ionasz, Alexander Schepsky, Jade Viarigi, Indridi Einar Reynisson, Vivian Pogenberg, Matthias Wilmanns, Margret Helga Ogmundsdottir, Eirikur Steingrimsson