Structure-activity relationship, biological, and pharmacological characterization of the proline sulfonamide ACT-462206: a potent, brain-penetrant dual orexin 1/orexin 2 receptor antagonist
脯氨酰磺酰胺 ACT-462206 的构效关系、生物学和药理学表征:一种强效的脑渗透性双食欲素 1/食欲素 2 受体拮抗剂
期刊:ChemMedChem
影响因子:3.6
doi:10.1002/cmdc.201402258
Christoph Boss, Catherine Roch-Brisbare, Michel A Steiner, Alexander Treiber, Hendrik Dietrich, Francois Jenck, Markus von Raumer, Thierry Sifferlen, Christine Brotschi, Bibia Heidmann, Jodi T Williams, Hamed Aissaoui, Romain Siegrist, John Gatfield