日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rational design of phenyl 2,4,5-trichlorobenzenesulfonate based thiosemicarbazones as α-glucosidase and α-amylase inhibitors: integrating enzymatic evaluation and molecular modeling

基于苯基2,4,5-三氯苯磺酸酯的硫代氨基脲类化合物作为α-葡萄糖苷酶和α-淀粉酶抑制剂的合理设计:酶学评价与分子建模的整合

Noreen, Faiqa; Zaki, Magdi E A; Sadeghian, Nastaran; Tokali, Feyzi Sinan; Taslimi, Parham; Alharthy, Rima D; Şenol, Halil; Zhao, Xianliang; Çakır, Furkan; Gomha, Sobhi M; Shafiq, Zahid

Synthesis and biological evaluation of 6-hydroxychromone based thiosemicarbazones as potential antidiabetic and antioxidant agents

6-羟基色酮基硫代氨基脲类化合物的合成及生物学评价:作为潜在的抗糖尿病和抗氧化剂

Zareen, Wajeeha; Ahmed, Nadeem; Siddique, Farhan; Taslimi, Parham; Khan, Muhammad Ali; Islam, Talha; Ismail, Mostafa A; Al-Rashida, Mariya; Zaki, Magdi E A; Gomha, Sobhi M; Alharthy, Rima D; Shafiq, Zahid

Design, Synthesis, In Vitro, and In Silico Studies of 5-(Diethylamino)-2-Formylphenyl Naphthalene-2-Sulfonate Based Thiosemicarbazones as Potent Anti-Alzheimer Agents.

5-(二乙氨基)-2-甲酰基苯基萘-2-磺酸酯基硫代氨基脲类化合物作为强效抗阿尔茨海默病药物的设计、合成、体外和计算机模拟研究

Farooq Urva, Islam Muhammad, Batool Zahra, Mali Suraj N, Jawarkar Rahul D, Gurav Shailesh S, Alharthy Rima D, Şenol Halil, Sadeghian Nastaran, Taslimi Parham, Shafiq Zahid, Schenone Silvia

Binding selectivity analysis of AURKs inhibitors through molecular dynamics simulation studies

通过分子动力学模拟研究分析AURK抑制剂的结合选择性

Alharthy, Rima D; Fatima, Ghulam; Yousaf, Numan; Iqbal, Muhammad Shaheen; Sattar, Sadia; Alanzi, Abdullah R; Ali, Ijaz; Muddassar, Muhammad

Identification of human phosphoglycerate mutase 1 (PGAM1) inhibitors using hybrid virtual screening approaches

利用混合虚拟筛选方法鉴定人磷酸甘油酸变位酶1 (PGAM1) 抑制剂

Yousaf, Numan; Alharthy, Rima D; Maryam; Kamal, Iqra; Saleem, Muhammad; Muddassar, Muhammad

Synthesis, Biological Evaluation, and Molecular Dynamics of Carbothioamides Derivatives as Carbonic Anhydrase II and 15-Lipoxygenase Inhibitors

合成、生物学评价及作为碳酸酐酶II和15-脂氧合酶抑制剂的硫代甲酰胺衍生物的分子动力学研究

Channar, Pervaiz Ali; Alharthy, Rima D; Ejaz, Syeda Abida; Saeed, Aamer; Iqbal, Jamshed

Investigations of Structural Requirements for BRD4 Inhibitors through Ligand- and Structure-Based 3D QSAR Approaches

通过基于配体和结构的3D QSAR方法研究BRD4抑制剂的结构要求

Tahir, Adeena; Alharthy, Rima D; Naseem, Saadia; Mahmood, Natasha; Ahmed, Mahmood; Shahzad, Khuram; Akhtar, Malik Nadeem; Hameed, Abdul; Sadiq, Irfan; Nawaz, Haq; Muddassar, Muhammad

N-Alkylated 1,4-Diazabicyclo[2.2.2]octane-Polyethylene Glycol Melt as Deep Eutectic Solvent for the Synthesis of Fisher Indoles and 1H-Tetrazoles

N-烷基化1,4-二氮杂双环[2.2.2]辛烷-聚乙二醇熔体作为低共熔溶剂用于合成费歇尔吲哚和1H-四唑

Ali Ghumro, Sarfaraz; Alharthy, Rima D; Al-Rashida, Mariya; Ahmed, Shakil; Malik, Muhammad Imran; Hameed, Abdul

Synthesis of triazole-linked morpholino oligonucleotides via Cu(I) catalysed cycloaddition

通过Cu(I)催化的环加成反应合成三唑连接的吗啉代寡核苷酸

Palframan, Matthew J; Alharthy, Rima D; Powalowska, Paulina K; Hayes, Christopher J