日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Evaluation of Malaria Parasite Transmission Competency Using a Nanozyme-Based Immunodiagnostic Targeting Female Gamete Antigen Release

利用基于纳米酶的免疫诊断方法靶向雌性配子抗原释放评估疟原虫的传播能力

Haghighi, Tabasom; Najer, Adrian; Broto, Marta; Dahalan, Farah A; Churchyard, Alisje; Yahiya, Sabrina; Famodimu, Mufuliat T; Tunnicliff, Mark; Abdelwahed, Aida; Tachibana, Mayumi; Ishino, Tomoko; Aniweh, Yaw; Awandare, Gordon A; Mahamar, Almahamoudou; Vanheer, Leen N; Bousema, Teun; Drakeley, Chris; Dicko, Alassane; Stone, William; Baum, Jake; Stevens, Molly M

Optimization and Characterization of N-Acetamide Indoles as Antimalarials That Target PfATP4

优化和表征靶向 PfATP4 的 N-乙酰胺吲哚类抗疟药

Awalt, Jon Kyle; Ooi, Zi Kang; Ashton, Trent D; Mansouri, Mahta; Calic, Petar P S; Zhou, Qingmiao; Vasanthan, Santhya; Lee, Serena; Loi, Katie; Jarman, Kate E; Penington, Jocelyn S; Qiu, Deyun; Zhang, Xinxin; Lehane, Adele M; Mao, Emma Y; Gancheva, Maria R; Wilson, Danny W; Giannangelo, Carlo; MacRaild, Christopher A; Creek, Darren J; Yeo, Tomas; Sheth, Tanaya; Fidock, David A; Churchyard, Alisje; Baum, Jake; Famodimu, Mufuliat T; Delves, Michael J; Kristan, Mojca; Stewart, Lindsay; Sutherland, Colin J; Coyle, Rachael; Jagoe, Hannah; Lee, Marcus C S; Chowdury, Mrittika; de Koning-Ward, Tania F; Baud, Delphine; Brand, Stephen; Jackson, Paul F; Cowman, Alan F; Dans, Madeline G; Sleebs, Brad E

Exploration and characterization of the antimalarial activity of cyclopropyl carboxamides that target the mitochondrial protein, cytochrome b

探索和表征靶向线粒体蛋白细胞色素b的环丙基羧酰胺类化合物的抗疟活性

Awalt, Jon Kyle; Su, Wenyin; Nguyen, William; Loi, Katie; Jarman, Kate E; Penington, Jocelyn S; Ramesh, Saishyam; Fairhurst, Kate J; Yeo, Tomas; Park, Heekuk; Uhlemann, Anne-Catrin; Chandra Maity, Bikash; De, Nirupam; Mukherjee, Partha; Chakraborty, Arnish; Churchyard, Alisje; Famodimu, Mufuliat T; Delves, Michael J; Baum, Jake; Mittal, Nimisha; Winzeler, Elizabeth A; Papenfuss, Anthony T; Chowdury, Mrittika; de Koning-Ward, Tania F; Maier, Alexander G; van Dooren, Giel G; Baud, Delphine; Brand, Stephen; Fidock, David A; Jackson, Paul F; Cowman, Alan F; Dans, Madeline G; Sleebs, Brad E

Optimization of 2,3-Dihydroquinazolinone-3-carboxamides as Antimalarials Targeting PfATP4

优化 2,3-二氢喹唑啉酮-3-甲酰胺类化合物作为靶向 PfATP4 的抗疟药

Ashton, Trent D; Dans, Madeline G; Favuzza, Paola; Ngo, Anna; Lehane, Adele M; Zhang, Xinxin; Qiu, Deyun; Chandra Maity, Bikash; De, Nirupam; Schindler, Kyra A; Yeo, Tomas; Park, Heekuk; Uhlemann, Anne-Catrin; Churchyard, Alisje; Baum, Jake; Fidock, David A; Jarman, Kate E; Lowes, Kym N; Baud, Delphine; Brand, Stephen; Jackson, Paul F; Cowman, Alan F; Sleebs, Brad E

Fast-Killing Tyrosine Amide ((S)-SW228703) with Blood- and Liver-Stage Antimalarial Activity Associated with the Cyclic Amine Resistance Locus (PfCARL)

快速杀灭酪氨酸酰胺((S)-SW228703)具有血液期和肝脏期抗疟活性,与环胺抗性基因座(PfCARL)相关

Imlay, Leah S; Lawong, Aloysus K; Gahalawat, Suraksha; Kumar, Ashwani; Xing, Chao; Mittal, Nimisha; Wittlin, Sergio; Churchyard, Alisje; Niederstrasser, Hanspeter; Crespo-Fernandez, Benigno; Posner, Bruce A; Gamo, Francisco-Javier; Baum, Jake; Winzeler, Elizabeth A; Laleu, Benoît; Ready, Joseph M; Phillips, Margaret A

Reaction hijacking of tyrosine tRNA synthetase as a new whole-of-life-cycle antimalarial strategy

酪氨酸tRNA合成酶的反应劫持作为一种新的全生命周期抗疟策略

Xie, Stanley C; Metcalfe, Riley D; Dunn, Elyse; Morton, Craig J; Huang, Shih-Chung; Puhalovich, Tanya; Du, Yawei; Wittlin, Sergio; Nie, Shuai; Luth, Madeline R; Ma, Liting; Kim, Mi-Sook; Pasaje, Charisse Flerida A; Kumpornsin, Krittikorn; Giannangelo, Carlo; Houghton, Fiona J; Churchyard, Alisje; Famodimu, Mufuliat T; Barry, Daniel C; Gillett, David L; Dey, Sumanta; Kosasih, Clara C; Newman, William; Niles, Jacquin C; Lee, Marcus C S; Baum, Jake; Ottilie, Sabine; Winzeler, Elizabeth A; Creek, Darren J; Williamson, Nicholas; Parker, Michael W; Brand, Stephen; Langston, Steven P; Dick, Lawrence R; Griffin, Michael D W; Gould, Alexandra E; Tilley, Leann

Live-cell fluorescence imaging of microgametogenesis in the human malaria parasite Plasmodium falciparum

人类疟原虫恶性疟原虫微配子发生的活细胞荧光成像

Sabrina Yahiya, Sarah Jordan, Holly X Smith, David C A Gaboriau, Mufuliat T Famodimu, Farah A Dahalan, Alisje Churchyard, George W Ashdown, Jake Baum

Design of proteasome inhibitors with oral efficacy in vivo against Plasmodium falciparum and selectivity over the human proteasome

设计对恶性疟原虫具有体内口服疗效且对人蛋白酶体具有选择性的蛋白酶体抑制剂

Xie, Stanley C; Metcalfe, Riley D; Mizutani, Hirotake; Puhalovich, Tanya; Hanssen, Eric; Morton, Craig J; Du, Yawei; Dogovski, Con; Huang, Shih-Chung; Ciavarri, Jeffrey; Hales, Paul; Griffin, Robert J; Cohen, Lawrence H; Chuang, Bei-Ching; Wittlin, Sergio; Deni, Ioanna; Yeo, Tomas; Ward, Kurt E; Barry, Daniel C; Liu, Boyin; Gillett, David L; Crespo-Fernandez, Benigno F; Ottilie, Sabine; Mittal, Nimisha; Churchyard, Alisje; Ferguson, Daniel; Aguiar, Anna Caroline C; Guido, Rafael V C; Baum, Jake; Hanson, Kirsten K; Winzeler, Elizabeth A; Gamo, Francisco-Javier; Fidock, David A; Baud, Delphine; Parker, Michael W; Brand, Stephen; Dick, Lawrence R; Griffin, Michael D W; Gould, Alexandra E; Tilley, Leann