Discovery of Imidazopyridines as Potent Inhibitors of Indoleamine 2,3-Dioxygenase 1 for Cancer Immunotherapy
发现咪唑并吡啶类化合物是吲哚胺2,3-双加氧酶1的强效抑制剂,可用于癌症免疫治疗
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.1c00014
Zhang, Liping; Cherney, Emily C; Zhu, Xiao; Lin, Tai-An; Gullo-Brown, Johnni; Maley, Derrick; Johnston-Allegretto, Kathy; Kopcho, Lisa; Fereshteh, Mark; Huang, Christine; Li, Xin; Traeger, Sarah C; Dhar, Gopal; Anandam, Aravind; Mahankali, Sandeep; Padmanabhan, Shweta; Rajanna, Prabhakar; Murali, Venkata; Mariappan, Thanga; Borzilleri, Robert; Vite, Gregory; Hunt, John T; Balog, Aaron