Freezing the Bioactive Conformation to Boost Potency: The Identification of BAY 85-8501, a Selective and Potent Inhibitor of Human Neutrophil Elastase for Pulmonary Diseases
冷冻生物活性构象以增强效力:鉴定 BAY 85-8501,一种用于治疗肺部疾病的选择性强效人中性粒细胞弹性蛋白酶抑制剂
期刊:ChemMedChem
影响因子:3.6
doi:10.1002/cmdc.201500131
Franz von Nussbaum, Volkhart M-J Li, Swen Allerheiligen, Sonja Anlauf, Lars Bärfacker, Martin Bechem, Martina Delbeck, Mary F Fitzgerald, Michael Gerisch, Heike Gielen-Haertwig, Helmut Haning, Dagmar Karthaus, Dieter Lang, Klemens Lustig, Daniel Meibom, Joachim Mittendorf, Ulrich Rosentreter, Martin