Stereospecific Resistance to N2-Acyl Tetrahydro-β-carboline Antimalarials Is Mediated by a PfMDR1 Mutation That Confers Collateral Drug Sensitivity
对N2-酰基四氢-β-咔啉类抗疟药的立体特异性耐药性是由PfMDR1突变介导的,该突变赋予了药物的附带敏感性。
期刊:ACS Infectious Diseases
影响因子:3.8
doi:10.1021/acsinfecdis.4c01001
Bremers, Emily K; Butler, Joshua H; Do Amaral, Leticia S; Merino, Emilio F; Almolhim, Hanan; Zhou, Bo; Baptista, Rodrigo P; Totrov, Maxim; Carlier, Paul R; Cassera, Maria Belen