日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

REV1 inhibition enhances trinucleotide repeat mutagenesis

REV1抑制增强三核苷酸重复序列突变

Siegel, Ava; Almstead, Daniel; Kothandaraman, Naveen; Reich, Jessica; Lamkin, Erica; Victor, Josh A; Grover, Aarzoo; Ikeh, Kanayo; Koval, Hannah; Crompton, Andrew; Jang, Hongjun; Lee, Hyejin; Del Rio Guerra, Roxana; Korzhnev, Dmitry M; Kyle Hadden, M; Hong, Jiyong; Zhou, Pei; Chatterjee, Nimrat

Single-Dose Anti-PD-L1/IL-15 Fusion Protein KD033 Generates Synergistic Antitumor Immunity with Robust Tumor-Immune Gene Signatures and Memory Responses

单剂量抗 PD-L1/IL-15 融合蛋白 KD033 产生协同抗肿瘤免疫力,并具有强大的肿瘤免疫基因特征和记忆反应

Stella A Martomo, Dan Lu, Zhanna Polonskaya, Xenia Luna, Zhikai Zhang, Sam Feldstein, Radovan Lumban-Tobing, Danielle K Almstead, Faical Miyara, Jeegar Patel

In vitro metabolism, reaction phenotyping, enzyme kinetics, CYP inhibition and induction potential of ataluren

Ataluren 的体外代谢、反应表型、酶动力学、CYP 抑制和诱导潜力

Ronald Kong, Jiyuan Ma, Seongwoo Hwang, Young-Choon Moon, Ellen M Welch, Marla Weetall, Joseph M Colacino, Neil Almstead, John Babiak, Elizabeth Goodwin

Ataluren Pharmacokinetics in Healthy Japanese and Caucasian Subjects

阿塔卢伦在健康日本人和白种人受试者中的药代动力学

Kong, Ronald; Laskin, Oscar L; Kaushik, Diksha; Jin, Fengbin; Ma, Jiyuan; McIntosh, Joseph; Souza, Marcio; Almstead, Neil

Oxy-Allyl Cation Catalysis: An Enantioselective Electrophilic Activation Mode

氧烯丙基阳离子催化:一种对映选择性亲电活化模式

Liu, Chun; Oblak, E Zachary; Vander Wal, Mark N; Dilger, Andrew K; Almstead, Danielle K; MacMillan, David W C

Phase 1 Study of Safety, Tolerability, and Pharmacokinetics of PTC299, an Inhibitor of Stress-Regulated Protein Translation

应激调节蛋白翻译抑制剂 PTC299 的安全性、耐受性和药代动力学 1 期研究

Marla Weetall, Thomas Davis, Gary Elfring, Valerie Northcutt, Liangxian Cao, Young-Choon Moon, Peter Riebling, Mandar Dali, Samit Hirawat, John Babiak, Joseph Colacino, Neil Almstead, Robert Spiegel, Stuart W Peltz

Identification of PTC725, an orally bioavailable small molecule that selectively targets the hepatitis C Virus NS4B protein

鉴定 PTC725,一种口服生物可利用的小分子,可选择性靶向丙型肝炎病毒 NS4B 蛋白

Zhengxian Gu, Jason D Graci, Frederick C Lahser, Jamie J Breslin, Stephen P Jung, James H Crona, Patricia McMonagle, Ellen Xia, Shaotang Liu, Gary Karp, Jin Zhu, Song Huang, Amin Nomeir, Marla Weetall, Neil G Almstead, Stuart W Peltz, Xiao Tong, Robert Ralston, Joseph M Colacino

Inhibition of U snRNP assembly by a virus-encoded proteinase

病毒编码蛋白酶对U snRNP组装的抑制作用

Almstead, Laura L; Sarnow, Peter