日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Organoselenium-based Schiff bases and amidic acid derivatives as promising anticancer agents targeting breast cancer by downregulating BCL-2: design, synthesis, and biological evaluation

基于有机硒的席夫碱和酰胺酸衍生物作为靶向乳腺癌、通过下调BCL-2表达的潜在抗癌药物:设计、合成和生物学评价

Shaaban, Saad; Hawas, Samia S; Elsharif, Asma M; Sharaky, Marwa; Ba-Ghazal, Hussein; Alaasar, Mohamed; Alatawi, Fatema S; Alomari, Khadra B; Eissa, Mohamed E; Al Khatib, Arwa Omar; Alnajjar, Radwan; Al-Karmalawy, Ahmed A

Targeted synthesis of a trimethoxyphenyltetrahydropyrimidine analogue designed as a DNA intercalator: in silico, multi-spectroscopic, thermodynamic, and in vitro approaches

以DNA嵌入剂为设计目标的三甲氧基苯基四氢嘧啶类似物的靶向合成:计算机模拟、多光谱学、热力学和体外方法

Al-Karmalawy, Ahmed A; Elmaaty, Ayman Abo; Magdy, Galal; Radwan, Aya Saad; Alnajjar, Radwan; Shaldam, Moataz A; Al Khatib, Arwa Omar; Almujri, Salem Salman; Abdullah Alzahrani, Abdullah Yahya; Tawfik, Haytham O

An in-depth study of indolone derivatives as potential lung cancer treatment

对吲哚酮衍生物作为潜在肺癌治疗药物的深入研究

Er-Rajy, Mohammed; El Fadili, Mohamed; Alnajjar, Radwan; Zarougui, Sara; Mujwar, Somdutt; Azzaoui, Khalil; Abuelizz, Hatem A; Hammouti, Belkheir; Elhallaoui, Menana

Discovery of natural scaffolds as HER2 inhibitors for breast cancer: virtual screening, molecular dynamics, and biological characterization with selectivity profiling.

发现天然支架作为乳腺癌 HER2 抑制剂:虚拟筛选、分子动力学和选择性分析的生物学表征

Hossam Asmaa, Abdallah Ingy I, El-Sebakhy Nadia A, Alnajjar Radwan, Mohyeldin Mohamed M

Donepezil-based rational design of N-substituted quinazolinthioacetamide candidates as potential acetylcholine esterase inhibitors for the treatment of Alzheimer's disease: in vitro and in vivo studies

基于多奈哌齐的N-取代喹唑啉硫代乙酰胺类化合物的合理设计:作为治疗阿尔茨海默病的潜在乙酰胆碱酯酶抑制剂:体外和体内研究

Al-Karmalawy, Ahmed A; Mohamed, Ahmed F; Shalaby, Heba Nasr; Elmaaty, Ayman Abo; El-Shiekh, Riham A; Zeidan, Mohamed A; Alnajjar, Radwan; Alzahrani, Abdullah Yahya Abdullah; Al Mughram, Mohammed H; Shaldam, Moataz A; Tawfik, Haytham O

Identification of Ureidocoumarin-Based Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors via Drug Repurposing Approach, Biological Evaluation, and In Silico Studies

通过药物重定位、生物学评价和计算机模拟研究鉴定脲基香豆素类选择性盘状结构域受体1 (DDR1) 抑制剂

El-Damasy, Ashraf K; Kim, Hyun Ji; Al-Karmalawy, Ahmed A; Alnajjar, Radwan; Khalifa, Mohamed M; Bang, Eun-Kyoung; Keum, Gyochang

Nuciferol C, a new sesquineolignan dimer from Cocos nucifera L.: bioactivity and theoretical investigation

椰子(Cocos nucifera L.)中一种新的倍半木脂素二聚体——Nuciferol C:生物活性及理论研究

Elsbaey, Marwa; Igarashi, Yasuhiro; Alnajjar, Radwan; Darwish, Khaled M; Miyamoto, Tomofumi

Investigating the anti-inflammatory potential of N-amidic acid organoselenium candidates: biological assessments, molecular docking, and molecular dynamics simulations

研究N-酰胺酸有机硒候选物的抗炎潜力:生物学评价、分子对接和分子动力学模拟

Althikrallah, Hanan A; Shaaban, Saad; Elmaaty, Ayman Abo; Ba-Ghazal, Hussein; Almarri, Mohammed N; Sharaky, Marwa; Alnajjar, Radwan; Al-Karmalawy, Ahmed A

Biological and computational assessments of thiazole derivative-reinforced bile salt enriched nano carriers: a new gate in targeting SARS-CoV-2 spike protein

噻唑衍生物增强型胆盐富集纳米载体的生物学和计算评估:靶向SARS-CoV-2刺突蛋白的新途径

Zakaria, Mohamed Y; Elmaaty, Ayman Abo; El-Shesheny, Rabeh; Alnajjar, Radwan; Kutkat, Omnia; Ben Moussa, Sana; Abdullah Alzahrani, Abdullah Yahya; El-Zahaby, Sally A; Al-Karmalawy, Ahmed A

Computational insights into rational design and virtual screening of pyrazolopyrimidine derivatives targeting Janus kinase 3 (JAK3)

利用计算方法对靶向 Janus 激酶 3 (JAK3) 的吡唑并嘧啶衍生物进行合理设计和虚拟筛选

Faris, Abdelmoujoud; Cacciatore, Ivana; Alnajjar, Radwan; Aouidate, Adnane; Al Mughram, Mohammed H; Elhallaoui, Menana