日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Piperazine ring toxicity in three novel anti-breast cancer drugs: an in silico and in vitro metabolic bioactivation approach using olaparib as a case study

三种新型抗乳腺癌药物中的哌嗪环毒性:以奥拉帕尼为例的计算机模拟和体外代谢生物活化方法

Thamer A Alsubi, Mohamed W Attwa, Hany W Darwish, Hatem A Abuelizz, Adnan A Kadi

In silico and in vitro metabolism of ribociclib: a mass spectrometric approach to bioactivation pathway elucidation and metabolite profiling

利用质谱法解析ribociclib的生物活化途径和代谢物谱,进行计算机模拟和体外代谢研究。

Alsubi, Thamer A; Attwa, Mohamed W; Bakheit, Ahmed H; Darwish, Hany W; Abuelizz, Hatem A; Kadi, Adnan A

Identification of reactive intermediate formation and bioactivation pathways in Abemaciclib metabolism by LC-MS/MS: in vitro metabolic investigation

通过 LC-MS/MS 鉴定 Abemaciclib 代谢中的反应中间体形成和生物活化途径:体外代谢研究

Adnan A Kadi, Hany W Darwish, Hatem A Abuelizz, Thamer A Alsubi, Mohamed W Attwa