日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Microglial-Targeted GCPII Inhibition Reverses Neurocognitive Impairment and Synaptic Loss After EcoHIV Infection.

靶向小胶质细胞的 GCPII 抑制可逆转 EcoHIV 感染后的神经认知障碍和突触丢失。

Zheng Yuxin, Huang Meixiang, Maragakis R Michael, Pietri Peter, Su Yu, Alt Jesse, Tenora Lukáš, Liyanage Wathsala, Wu Ying, Thomas Mary-Anne, Kannan Rangaramanujam M, Zhu Xiaolei, Rais Rana, Slusher Barbara S

Targeting NAAG metabolism restores cognition and synaptic integrity in EcoHIV-infected mice

靶向NAAG代谢可恢复EcoHIV感染小鼠的认知功能和突触完整性。

Zheng, Yuxin; Huang, Meixiang; Maragakis, R Michael; Pietri, Peter; Su, Yu; Alt, Jesse; Wu, Ying; Finney, Colin; Peters, Diane E; Zhu, Xiaolei; Rais, Rana; Slusher, Barbara S

Translin deletion impairs cocaine-induced locomotor sensitization and RGS8 expression in the nucleus accumbens

Translin基因缺失会损害伏隔核中可卡因诱导的运动敏化和RGS8表达。

Fu, Xiu-Ping; Wu, Ren-Kun; Shah, Aparna P; Ladenheim, Bruce; Alt, Jesse; Cadet, Jean Lud; Rais, Rana; Chandra, Ramesh; Cen, Xiao-Bo; Baraban, Jay M

Mass spectrometry-guided discovery of novel GCPII inhibitor scaffolds

质谱引导下新型GCPII抑制剂骨架的发现

Wiseman, Robyn; Thomas, Ajit G; Janiszewski, John; Hoxie, Nate; Lee, Chae Bin; Wu, Ying; Tsukamoto, Takashi; Ye, Lin; Ronzetti, Michael; Shrimp, Jonathan H; Adderley, Davina; Rai, Ganesha; Rais, Rana; Alt, Jesse; Hall, Matthew D; Hu, Xin; Kales, Stephen C; Slusher, Barbara S

The SWELL1 Channel Promotes Ischemic Brain Damage by Mediating Neuronal Swelling and Glutamate Toxicity

SWELL1通道通过介导神经元肿胀和谷氨酸毒性促进缺血性脑损伤

Chen, Jianan; Yang, Junhua; Chu, Jiachen; Chen, Kevin Hong; Alt, Jesse; Rais, Rana; Qiu, Zhaozhu

Pharmacokinetic Evaluation of Neutral Sphinghomyelinase2 (nSMase2) Inhibitor Prodrugs in Mice and Dogs

中性鞘磷脂酶2 (nSMase2) 抑制剂前药在小鼠和犬体内的药代动力学评价

Ranjit, Arina; Lee, Chae Bin; Tenora, Lukáš; Mettu, Vijaya Saradhi; Pal, Arindom; Alt, Jesse; Slusher, Barbara S; Rais, Rana

Neutral sphingomyelinase 2 inhibitors based on the pyrazolo[1,5-a]pyrimidin-3-amine scaffold

基于吡唑并[1,5-a]嘧啶-3-胺骨架的中性鞘磷脂酶2抑制剂

Novotna, Katerina; Thomas, Ajit G; Stepanek, Ondrej; Murphy, Brennan; Hin, Niyada; Skacel, Jan; Mueller, Louis; Tenora, Lukas; Pal, Arindom; Alt, Jesse; Wu, Ying; Paule, James; Rais, Rana; Slusher, Barbara S; Tsukamoto, Takashi

Topical SCD-153, a 4-methyl itaconate prodrug, for the treatment of alopecia areata

局部用药 SCD-153,一种 4-甲基衣康酸前药,用于治疗斑秃

Tsai, Jerry; Gori, Sadakatali; Alt, Jesse; Tiwari, Sandhya; Iyer, Jitesh; Talwar, Rashmi; Hinsu, Denish; Ahirwar, Kailash; Mohanty, Swayam; Khunt, Chintan; Sutariya, Brijesh; Jani, Kaushal; Venkatasubbaiah, Venkatesha; Patel, Ashok; Meghapara, Jasmin; Joshi, Kaushal; Sahu, Rajanikanta; Rana, Vijay; Nigade, Prashant; Talluri, Ravi S; Murty, Kadiyala V S N; Joshi, Kiritkumar; Ramanathan, Vikram; Li, Ang; Islam, Nasif; Snajdr, Ivan; Majer, Pavel; Rais, Rana; Slusher, Barbara S; Garza, Luis A

Discovery of DRP-104, a tumor-targeted metabolic inhibitor prodrug

发现肿瘤靶向代谢抑制剂前药DRP-104

Rais, Rana; Lemberg, Kathryn M; Tenora, Lukáš; Arwood, Matthew L; Pal, Arindom; Alt, Jesse; Wu, Ying; Lam, Jenny; Aguilar, Joanna Marie H; Zhao, Liang; Peters, Diane E; Tallon, Carolyn; Pandey, Rajeev; Thomas, Ajit G; Dash, Ranjeet P; Seiwert, Tanguy; Majer, Pavel; Leone, Robert D; Powell, Jonathan D; Slusher, Barbara S

Thieno[2,3-d]pyrimidine-Based Positive Allosteric Modulators of Human Mas-Related G Protein-Coupled Receptor X1 (MRGPRX1)

基于噻吩并[2,3-d]嘧啶的人类Mas相关G蛋白偶联受体X1(MRGPRX1)正向变构调节剂

Berhane, Ilyas; Hin, Niyada; Thomas, Ajit G; Huang, Qian; Zhang, Chi; Veeravalli, Vijayabhaskar; Wu, Ying; Ng, Justin; Alt, Jesse; Rojas, Camilo; Hihara, Hiroe; Aoki, Mika; Yoshizawa, Kyoko; Nishioka, Tomoki; Suzuki, Shuichi; He, Shao-Qiu; Peng, Qi; Guan, Yun; Dong, Xinzhong; Raja, Srinivasa N; Slusher, Barbara S; Rais, Rana; Tsukamoto, Takashi