Identification of 5-(Aryl/Heteroaryl)amino-4-quinolones as Potent Membrane-Disrupting Agents to Combat Antibiotic-Resistant Gram-Positive Bacteria
鉴定 5-(芳基/杂芳基)氨基-4-喹诺酮类化合物为有效膜破坏剂,可对抗抗生素耐药性革兰氏阳性菌
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.2c01151
John R Schultz, Stephen K Costa, Gorakhnath R Jachak, Pooja Hegde, Matthew Zimmerman, Yan Pan, Michaele Josten, Chinedu Ejeh, Travis Hammerstad, Hans Georg Sahl, Pedro M Pereira, Mariana G Pinho, Véronique Dartois, Ambrose Cheung, Courtney C Aldrich