日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

(N)-Methanocarba Adenosine Derivatives as Dual Modulators of P-Glycoprotein and ABCG2 Transporters

(N)-甲氧基碳腺苷衍生物作为P-糖蛋白和ABCG2转运蛋白的双重调节剂

Murakami, Megumi; Tosh, Dilip K; Salazar, Paula B; Jacobson, Kenneth A; Ambudkar, Suresh V

Nanoengineered photosensitizers for photodynamic priming to overcome P-glycoprotein-mediated multidrug resistance.

利用纳米工程光敏剂进行光动力启动,以克服 P-糖蛋白介导的多药耐药性。

Rahman Idrisa, Meda Anju, Moore Kaitlyn A, Srivastava Payal, Dasgupta Anika, Sajid Andaleeb, Ambudkar Suresh V, Huang Huang-Chiao

Correction: Abcg2a is the functional homolog of human ABCG2 expressed at the zebrafish blood-brain barrier

更正:Abcg2a 是人类 ABCG2 的功能同源物,在斑马鱼血脑屏障处表达。

Thomas, Joanna R; Frye, William J E; Robey, Robert W; Warner, Andrew C; Butcher, Donna; Matta, Jennifer L; Morgan, Tamara C; Edmondson, Elijah F; Salazar, Paula B; Ambudkar, Suresh V; Gottesman, Michael M

Structure-activity relationship studies on 2-thienylidene substituted 3-oxo-2,3-dihydrobenzofuran-7-carboxamides as poly (ADP-ribose) polymerase inhibitors

2-噻吩亚甲基取代的3-氧代-2,3-二氢苯并呋喃-7-甲酰胺作为聚(ADP-核糖)聚合酶抑制剂的构效关系研究

Salami, Abosede; Adiele, Ugochi; Coate, Griffin; Diolaiti, Morgan; Chen, Huadong; Lu, Junhao; Ashworth, Alan; Patil, Manisha; Fleishman, Joshua S; Ramaraju, Andhavaram; Patel, Akanksha; Patel, Himaxi; Patel, Ketankumar; Murakami, Megumi; Ambudkar, Suresh V; Talele, Tanaji T

Conversion of Human Multidrug Transporter P-glycoprotein (ABCB1) from Drug Efflux to Uptake Pump: Evidence for a Switch Region Modulating the Direction of Substrate Transport

人多药转运蛋白P-糖蛋白(ABCB1)从药物外排泵向摄取泵的转化:调节底物转运方向的转换区证据

Sajid, Andaleeb; Ranganathan, Nandhini; Guha, Rajan; Murakami, Megumi; Ahmed, Shafaq; Durell, Stewart R; Ambudkar, Suresh V

Highly Sensitive Multiplexed Detection of Brain‐Derived Tau and Phosphorylated Tau Proteoforms with the NULISA Technology

利用NULISA技术对脑源性tau蛋白和磷酸化tau蛋白进行高灵敏度多重检测

Wang, Yi-Jun; Patel, Bhargav A; Anreddy, Nagaraju; Zhang, Yun-Kai; Zhang, Guan-Nan; Alqahtani, Saeed; Singh, Satyakam; Shukla, Suneet; Kaddoumi, Amal; Ambudkar, Suresh V; Talele, Tanaji T; Chen, Zhe-Sheng; Ma, Xiao‐Jun; Iyengar, Shweta; Deshmukh, Shalaka; Comandor, Roopa; Wang, Li; Kim, Sean; Xu, Xiaomei; Feng, Wei; Qiu, Xiaolei; Zhang, Bingqing; Luo, Yuling

Functional Implications of the Conformational Landscape of a Multidrug Transporter Revealed by Structures of Zebrafish Abcb4

斑马鱼Abcb4结构揭示多药转运蛋白构象图景的功能意义

Zhan, Jingyu; Hsieh, Chao-Ming; Esser, Lothar; Lang, Zabrina C; Morton, Abraham J; Robey, Robert; Zhou, Fei; Ambudkar, Suresh V; Huang, Rick K; Gottesman, Michael M; Xia, Di

Abcg2a is the functional homolog of human ABCG2 expressed at the zebrafish blood-brain barrier

Abcg2a是人类ABCG2的功能同源物,在斑马鱼血脑屏障处表达。

Thomas, Joanna R; Frye, William J E; Robey, Robert W; Warner, Andrew C; Butcher, Donna; Matta, Jennifer L; Morgan, Tamara C; Edmondson, Elijah F; Salazar, Paula B; Ambudkar, Suresh V; Gottesman, Michael M

Mutational analysis reveals the importance of residues of the access tunnel inhibitor site to human P-glycoprotein (ABCB1)-mediated transport

突变分析揭示了通道抑制位点残基对人P-糖蛋白(ABCB1)介导的转运的重要性

Salazar, Paula B; Murakami, Megumi; Ranganathan, Nandhini; Durell, Stewart R; Ambudkar, Suresh V

Magnolol derivatives as specific and noncytotoxic inhibitors of breast cancer resistance protein (BCRP/ABCG2)

木兰醇衍生物作为乳腺癌耐药蛋白(BCRP/ABCG2)的特异性无细胞毒性抑制剂

da Silva Zanzarini, Isadora; Henrique Kita, Diogo; Scheiffer, Gustavo; Karoline Dos Santos, Kelly; de Paula Dutra, Julia; Augusto Pastore, Matteo; Gomes de Moraes Rego, Fabiane; Picheth, Geraldo; Ambudkar, Suresh V; Pulvirenti, Luana; Cardullo, Nunzio; Rotuno Moure, Vivian; Muccilli, Vera; Tringali, Corrado; Valdameri, Glaucio