日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A3 adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity

含有多巴胺部分的 A3 腺苷受体激动剂可增强跨物种亲和力

Dilip K Tosh, Veronica Salmaso, Ryan G Campbell, Harsha Rao, Amelia Bitant, Eline Pottie, Christophe P Stove, Naili Liu, Oksana Gavrilova, Zhan-Guo Gao, John A Auchampach, Kenneth A Jacobson

Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A3 Adenosine Receptors: Affinity Enhancement by N6-(2-Phenylethyl) Substitution

截短的 (N)-亚甲基羰基核苷作为小鼠和人类 A3 腺苷受体的部分激动剂:通过 N6-(2-苯乙基) 取代增强亲和力

Dilip K Tosh, Veronica Salmaso, Harsha Rao, Amelia Bitant, Courtney L Fisher, David I Lieberman, Helmut Vorbrüggen, Marc L Reitman, Oksana Gavrilova, Zhan-Guo Gao, John A Auchampach, Kenneth A Jacobson

Structure activity relationship of 2-arylalkynyl-adenine derivatives as human A3 adenosine receptor antagonists

2-芳基炔基腺嘌呤衍生物作为人类 A3 腺苷受体拮抗剂的构效关系

Jinha Yu, Philip Mannes, Young-Hwan Jung, Antonella Ciancetta, Amelia Bitant, David I Lieberman, Sami Khaznadar, John A Auchampach, Zhan-Guo Gao, Kenneth A Jacobson