日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A cryptic pocket in CB1 drives peripheral and functional selectivity

CB1 中的一个隐蔽口袋驱动外周和功能选择性

Rangari, Vipin Ashok; O'Brien, Evan S; Powers, Alexander S; Slivicki, Richard A; Bertels, Zachariah; Appourchaux, Kevin; Aydin, Deniz; Ramos-Gonzalez, Nokomis; Mwirigi, Juliet; Lin, Li; Mangutov, Elizaveta; Sobecks, Briana L; Awad-Agbaria, Yaseen; Uphade, Manoj B; Aguilar, Jhoan; Peddada, Teja Nikhil; Shiimura, Yuki; Huang, Xi-Ping; Folarin-Hines, Jakayla; Payne, Maria; Kalathil, Anirudh; Varga, Balazs R; Kobilka, Brian K; Pradhan, Amynah A; Cameron, Michael D; Kumar, Kaavya Krishna; Dror, Ron O; Gereau, Robert W 4th; Majumdar, Susruta

Structure-guided design of partial agonists at an opioid receptor.

基于结构的阿片受体部分激动剂设计

Varga Balazs R, Bernhard Sarah M, El Daibani Amal, Zaidi Saheem A, Lam Jordy H, Aguilar Jhoan, Appourchaux Kevin, Nazarova Antonina L, Kouvelis Alexa, Shinouchi Ryosuke, Hammond Haylee R, Eans Shainnel O, Weinreb Violetta, Margolis Elyssa B, Fay Jonathan F, Huang Xi-Ping, Pradhan Amynah, Katritch Vsevolod, McLaughlin Jay P, Majumdar Susruta, Che Tao

Enhancement of the endocannabinoid system through monoacylglycerol lipase inhibition relieves migraine-associated pain in mice

通过抑制单酰甘油脂肪酶增强内源性大麻素系统可缓解小鼠偏头痛相关疼痛

Mangutov, Elizaveta; Awad-Igbaria, Yaseen; Siegersma, Kendra; Gastambide, Francois; Asuni, Ayodeji A; Pradhan, Amynah A A

Activation of δ-opioid receptors blocks allodynia in a model of headache induced by PACAP

δ-阿片受体的激活可阻断PACAP诱导的头痛模型中的痛觉过敏。

Mangutov, Elizaveta; Dripps, Isaac; Siegersma, Kendra; Zhang, Yanping; Bocian, Rebecca; Asif, Sarah; Halbesma, Timothy; Witkowski, Wiktor; Pradhan, Amynah A

Delta opioid receptors: Overlooked outlier or the next big thing

δ阿片受体:被忽视的异类还是下一个重大发现

El Daibani, Amal; Burgess, Gwendolyn; Rysztak, Lauren; Jutkiewicz, Emily; Pradhan, Amynah A

Evidence-based recommendations for diagnosing and managing dentine hypersensitivity in clinical practice: insights from the Middle East and Africa

基于循证医学的牙本质过敏症临床诊断和治疗建议:来自中东和非洲的启示

Cekici, Ali; Shaikh, Amynah; Alsayed, Arwa; Gokbuget, Aslan Yasar; Patel, Ebrahim; Marei, Hesham; Awad, Manal; Banday, Ninette; Habib, Nour A; Osailan, Samira M; Theuri, Tim; Adeyemi, Tope Emmanuel; Parkinson, Charlie R; Hamdy, Ahmed; Thomas, Juhi

Combination Targeted Therapy in Relapsed Diffuse Large B-Cell Lymphoma

复发性弥漫性大B细胞淋巴瘤的联合靶向治疗

Melani, Christopher; Lakhotia, Rahul; Pittaluga, Stefania; Phelan, James D; Huang, Da Wei; Wright, George; Simard, Jillian; Muppidi, Jagan; Thomas, Craig J; Ceribelli, Michele; Tosto, Frances A; Yang, Yandan; Xu, Weihong; Davies-Hill, Theresa; Pack, Svetlana D; Peer, Cody J; Arisa, Oluwatobi; Mena, Esther; Lindenberg, Liza; Bergvall, Ethan; Portell, Craig A; Farah, Rafic J; Lee, Seung Tae; Pradhan, Amynah; Morrison, Candis; Tadese, Atekelt; Juanitez, Anna Marie; Lu, Crystal; Jacob, Allison; Simmons, Heidi; Figg, William D; Steinberg, Seth M; Jaffe, Elaine S; Roschewski, Mark; Staudt, Louis M; Wilson, Wyndham H

Regulation of headache response and transcriptomic network by the trigeminal ganglion clock

三叉神经节时钟对头痛反应和转录组网络的调节

Chorong Han, Ji Ye Lim, Nobuya Koike, Sun Young Kim, Kaori Ono, Celia K Tran, Elizaveta Mangutov, Eunju Kim, Yanping Zhang, Lingyong Li, Amynah A Pradhan, Kazuhiro Yagita, Zheng Chen, Seung-Hee Yoo, Mark J Burish

Glial activation in pain and emotional processing regions in the nitroglycerin mouse model of chronic migraine

硝酸甘油诱导慢性偏头痛小鼠模型中疼痛和情绪处理区域的神经胶质细胞激活

Cropper, Haley C; Conway, Catherine M; Wyche, Whitney; Pradhan, Amynah A

Identification of 1,3,8-Triazaspiro[4.5]Decane-2,4-Dione Derivatives as a Novel δ Opioid Receptor-Selective Agonist Chemotype

鉴定出1,3,8-三氮杂螺[4.5]癸烷-2,4-二酮衍生物为一种新型δ阿片受体选择性激动剂化学型

Meqbil, Yazan J; Aguilar, Jhoan; Blaine, Arryn T; Chen, Lan; Cassell, Robert J; Pradhan, Amynah A; van Rijn, Richard M