日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A cryptic pocket in CB1 drives peripheral and functional selectivity

CB1 中的一个隐蔽口袋驱动外周和功能选择性

Rangari, Vipin Ashok; O'Brien, Evan S; Powers, Alexander S; Slivicki, Richard A; Bertels, Zachariah; Appourchaux, Kevin; Aydin, Deniz; Ramos-Gonzalez, Nokomis; Mwirigi, Juliet; Lin, Li; Mangutov, Elizaveta; Sobecks, Briana L; Awad-Agbaria, Yaseen; Uphade, Manoj B; Aguilar, Jhoan; Peddada, Teja Nikhil; Shiimura, Yuki; Huang, Xi-Ping; Folarin-Hines, Jakayla; Payne, Maria; Kalathil, Anirudh; Varga, Balazs R; Kobilka, Brian K; Pradhan, Amynah A; Cameron, Michael D; Kumar, Kaavya Krishna; Dror, Ron O; Gereau, Robert W 4th; Majumdar, Susruta

Enhancement of the endocannabinoid system through monoacylglycerol lipase inhibition relieves migraine-associated pain in mice

通过抑制单酰甘油脂肪酶增强内源性大麻素系统可缓解小鼠偏头痛相关疼痛

Mangutov, Elizaveta; Awad-Igbaria, Yaseen; Siegersma, Kendra; Gastambide, Francois; Asuni, Ayodeji A; Pradhan, Amynah A A

Activation of δ-opioid receptors blocks allodynia in a model of headache induced by PACAP

δ-阿片受体的激活可阻断PACAP诱导的头痛模型中的痛觉过敏。

Mangutov, Elizaveta; Dripps, Isaac; Siegersma, Kendra; Zhang, Yanping; Bocian, Rebecca; Asif, Sarah; Halbesma, Timothy; Witkowski, Wiktor; Pradhan, Amynah A

Delta opioid receptors: Overlooked outlier or the next big thing

δ阿片受体:被忽视的异类还是下一个重大发现

El Daibani, Amal; Burgess, Gwendolyn; Rysztak, Lauren; Jutkiewicz, Emily; Pradhan, Amynah A

Regulation of headache response and transcriptomic network by the trigeminal ganglion clock

三叉神经节时钟对头痛反应和转录组网络的调节

Chorong Han, Ji Ye Lim, Nobuya Koike, Sun Young Kim, Kaori Ono, Celia K Tran, Elizaveta Mangutov, Eunju Kim, Yanping Zhang, Lingyong Li, Amynah A Pradhan, Kazuhiro Yagita, Zheng Chen, Seung-Hee Yoo, Mark J Burish

Glial activation in pain and emotional processing regions in the nitroglycerin mouse model of chronic migraine

硝酸甘油诱导慢性偏头痛小鼠模型中疼痛和情绪处理区域的神经胶质细胞激活

Cropper, Haley C; Conway, Catherine M; Wyche, Whitney; Pradhan, Amynah A

Identification of 1,3,8-Triazaspiro[4.5]Decane-2,4-Dione Derivatives as a Novel δ Opioid Receptor-Selective Agonist Chemotype

鉴定出1,3,8-三氮杂螺[4.5]癸烷-2,4-二酮衍生物为一种新型δ阿片受体选择性激动剂化学型

Meqbil, Yazan J; Aguilar, Jhoan; Blaine, Arryn T; Chen, Lan; Cassell, Robert J; Pradhan, Amynah A; van Rijn, Richard M

PACAP-PAC1 receptor inhibition is effective in opioid induced hyperalgesia and medication overuse headache models

PACAP-PAC1 受体抑制对阿片类药物引起的痛觉过敏和药物过度使用性头痛模型有效

Zachariah Bertels, Elizaveta Mangutov, Kendra Siegersma, Haley C Cropper, Alycia Tipton, Amynah A Pradhan

Neuronal complexity is attenuated in preclinical models of migraine and restored by HDAC6 inhibition

偏头痛临床前模型中的神经元复杂性减弱,而 HDAC6 抑制可恢复神经元复杂性

Zachariah Bertels, Harinder Singh, Isaac Dripps, Kendra Siegersma, Alycia F Tipton, Wiktor D Witkowski, Zoie Sheets, Pal Shah, Catherine Conway, Elizaveta Mangutov, Mei Ao, Valentina Petukhova, Bhargava Karumudi, Pavel A Petukhov, Serapio M Baca, Mark M Rasenick, Amynah A Pradhan

Delta opioid receptor regulation of calcitonin gene-related peptide dynamics in the trigeminal complex

三叉神经复合体中δ阿片受体调节降钙素基因相关肽的动力学

Laura S Moye, Kendra Siegersma, Isaac Dripps, Wiktor Witkowski, Elizaveta Mangutov, Dong Wang, Grégory Scherrer, Amynah A Pradhan