日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting glycerophospholipid biosynthesis overcomes chemoresistance driven by SLFN11 loss in Ewing sarcoma

靶向甘油磷脂生物合成可克服尤文氏肉瘤中由SLFN11缺失引起的化疗耐药性

Chakraborty, Kasturee; Burman, Ritambhar; Satheesh, Saharsh; Kieffer, Matthew; Karuhatty, Chandni; Yuan, Zuo-Fei; Tan, Haiyan; Lkhagva, Ankhbayar; High, Anthony A; Wang, Xusheng; Refaat, Alaa; Twarog, Nathaniel R; Zhang, Weixing; Wang, Yaxu; Fan, Yiping; Li, Qian; Madan Babu, M; Shelat, Anang A; Stewart, Elizabeth; Dyer, Michael A; Bagga, Puneet

NanoBRET Tracer Development for Class I Bromodomain Target Engagement in Live Cells

用于活细胞中 I 类溴结构域靶标结合的 NanoBRET 示踪剂的开发

Sneddon, Molly S; Tsou, Chun-Ju; Fu, Xiang; Shelat, Anang A; Pomerantz, William C K

Prevalence of cyp51A variants in a US collection of Aspergillus fumigatus clinical isolates and comparative analysis of their contribution to triazole antifungal resistance

美国烟曲霉临床分离株中cyp51A变异体的流行情况及其对三唑类抗真菌药物耐药性贡献的比较分析

Gómez Londoño, Luisa Fernanda; Souza, Ana Camila Oliveira; Burt, Brooks; Das, Sourav; Ge, Wenbo; Meza-Perez, Vanessa; Wiederhold, Nathan P; Shelat, Anang A; Cuomo, Christina A; Fortwendel, Jarrod R; Rogers, P David

Targeting the p53 pathway to treat atypical teratoid rhabdoid tumors

靶向p53通路治疗非典型畸胎瘤样横纹肌瘤

Refaat, Alaa; Cho, Hyekyung P; Williams, Justin S; Stripay, Jennifer; Blankenship, Kaley; Mercer, Kimberly S; De Vries, Rebekah; Connelly, Michele; Ganguly, Debolina; Robinson, Sarah; Savage, Evan; Twarog, Nathaniel R; Attery, Ayush; Laha, Dipranjan; Yu, Kaiwen; Poudel, Suresh; Dhanda, Sandeep K; Stewart, Clinton F; Freeman, Burgess B; Roberts, Charles W M; Tinkle, Christopher; Stewart, Elizabeth A; Upadhyaya, Santhosh A; Shelat, Anang A; Roussel, Martine F

Genetic modeling of ELP1-associated Sonic hedgehog medulloblastoma identifies MDM2 as a selective therapeutic target

ELP1相关Sonic hedgehog髓母细胞瘤的遗传建模鉴定出MDM2为选择性治疗靶点

Shiekh Tanveer Ahmad ,Yiran Li ,Jesus Garcia-Lopez ,Brian L Gudenas ,Jennifer Hadley ,Leena Paul ,Stephanie C Wu ,Alaa Refaat ,Marija Kojic ,Melissa Batts ,Taha Soliman ,Aaron Pitre ,Frederik Arnskötter ,Frederique Zindy ,Alun Jones ,Nathaniel R Twarog ,Anand Mayasundari ,Brandon Bianski ,Christopher Tinkle ,Abbas Shirinifard ,Laura Janke ,Meifen Lu ,Sara A Lewis ,Arzu Onar-Thomas ,Stefan M Pfister ,Amar Gajjar ,Suzanne J Baker ,Martine F Roussel ,Zoran Rankovic ,Giles W Robinson ,Brent A Orr ,Brandon Wainwright ,Anang A Shelat ,Sebastian M Waszak ,Lena M Kutscher ,Hong Lin ,Paul A Northcott

A screen to identify antifungal antagonists reveals a variety of pharmacotherapies that induce echinocandin tolerance in Candida albicans

一项旨在识别抗真菌拮抗剂的筛选研究揭示了多种可诱导白色念珠菌产生棘白菌素耐受性的药物疗法。

Reitler, Parker; DeJarnette, Christian A; Kumar, Ravinder; Tucker, Katie M; Peters, Tracy L; Twarog, Nathaniel R; Shelat, Anang A; Palmer, Glen E

The Combination of PARP and Topoisomerase 1 Inhibitors Improves Radiation Therapy for Ewing Sarcoma

PARP抑制剂和拓扑异构酶1抑制剂联合应用可改善尤文氏肉瘤的放射治疗效果

Xie, Jia; Mellado-Lagarde, Marcia M; Blankenship, Kaley; Ganguly, Debolina; Twarog, Nathaniel R; Bianski, Brandon; Kieffer, Matthew; Atkinson, Stefan; Sheppard, Heather; Gartrell, Jessica; Cler, Samuel; Federico, Sara M; Stewart, Elizabeth A; Tinkle, Christopher L; Shelat, Anang A

Capmatinib is an effective treatment for MET-fusion driven pediatric high-grade glioma and synergizes with radiotherapy

卡马替尼是治疗MET融合基因驱动的儿童高级别胶质瘤的有效药物,并且与放射疗法具有协同作用。

Zuckermann, Marc; He, Chen; Andrews, Jared; Bagchi, Aditi; Sloan-Henry, Roketa; Bianski, Brandon; Xie, Jia; Wang, Yingzhe; Twarog, Nathaniel; Onar-Thomas, Arzu; Ernst, Kati J; Yang, Lei; Li, Yong; Zhu, Xiaoyan; Ocasio, Jennifer K; Budd, Kaitlin M; Dalton, James; Li, Xiaoyu; Chepyala, Divyabharathi; Zhang, Junyuan; Xu, Ke; Hover, Laura; Roach, Jordan T; Chan, Kenneth Chun-Ho; Hofmann, Nina; McKinnon, Peter J; Pfister, Stefan M; Shelat, Anang A; Rankovic, Zoran; Freeman, Burgess B 3rd; Chiang, Jason; Jones, David T W; Tinkle, Christopher L; Baker, Suzanne J

Combination of Ribociclib with BET-Bromodomain and PI3K/mTOR Inhibitors for Medulloblastoma Treatment In Vitro and In Vivo

体外和体内研究Ribociclib联合BET-溴结构域抑制剂和PI3K/mTOR抑制剂治疗髓母细胞瘤

Jonchere, Barbara; Williams, Justin; Zindy, Frederique; Liu, Jingjing; Robinson, Sarah; Farmer, Dana M; Min, Jaeki; Yang, Lei; Stripay, Jennifer L; Wang, Yingzhe; Freeman, Burgess B; Yu, Jiyang; Shelat, Anang A; Rankovic, Zoran; Roussel, Martine F

Fragment-Based NMR Screening of the BPTF PHD Finger Methyl Lysine Reader Leads to the First Small-Molecule Inhibitors

基于片段的 NMR 筛选 BPTF PHD 指状甲基赖氨酸读取蛋白,发现了首批小分子抑制剂

Buchholz, Caroline R; Sneddon, Molly S; McPherson, Joseph E; Das, Sourav; Gee, Clifford T; Grillo, Michael J; Chai, Sergio C; Lee, Richard E; Chen, Taosheng; Harki, Daniel A; Shelat, Anang A; Pomerantz, William C K