日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Drugging the intrinsically disordered transactivation domain of androgen receptor

药物靶向雄激素受体固有无序的转录激活结构域

Obst, Jon K; Banuelos, Carmen A; Jian, Kunzhong; Tien, Amy H; Shkrabak, Oleksandr A; Wang, Jun; Mawji, Nasrin R; Tam, Teresa; Vuckovic, Marija; Williams, David E; Rogalski, Jason C; Yuan, Xiaojing; Strynadka, Natalie C J; Andersen, Raymond J; Sadar, Marianne D

Identification and characterization of five anti-mitotic sesquiterpene lactones from Arnica cordifolia

从山金车中鉴定和表征五种抗有丝分裂倍半萜内酯

Lockwood, Tanner C; Williams, David E; Molina, Layla; Andersen, Raymond J; Golsteyn, Roy M

Vacuolar-ATPase inhibitors are antimicrobial agents active against intracellular mycobacteria

液泡ATPase抑制剂是具有抗细胞内分枝杆菌活性的抗菌剂。

Rankine-Wilson, Leah; Shapira, Tirosh; Felker, Jake; Christofferson, Matthew; Sahile, Henok; Chao, Joseph; Afshar, Houria; Andersen, Raymond J; Sun, Jim; Av-Gay, Yossef

NMR Analysis and Assignment of a Biosynthesis Gene Cluster for Trichokonins VI and VIII, Antiplasmodial Large Peptaibols Produced by a Trichoderma sp. Fungus

对木霉属真菌产生的抗疟原虫大肽类化合物——毛霉素VI和VIII的生物合成基因簇进行核磁共振分析和鉴定

Bertonha, Ariane F; Williams, David E; Nicacio, Karen J; de Amorim, Marcelo R; Schoellhorn, Sydney M; Aguiar, Anna Caroline C; Valdes, Talita Alvarenga; Mendes, Giovana Rossi; Moura, Igor M R; Michaliski, Lamonielli F; Gotha, Matheus; Zuccarino, Caue A W; Sette, Lara D; Ferreira, Antônio G; Andersen, Raymond J; Guido, Rafael Victorio Carvalho; Berlinck, Roberto G S

Phenotypic screening in influenza-infected zebrafish identifies Nrf2-mediated compound protective against ischemia-reperfusion injury.

对感染流感的斑马鱼进行表型筛选,发现 Nrf2 介导的化合物可保护其免受缺血再灌注损伤

Latreille Elyse, Mukkala Avinash Naraiah, Sanwal Rajiv, Yun Junghwa, Wei Kuiru, Petrut Raluca, Farahani Nikki Zamani, Philip Tristan, Xu Leo, Bateman Tom, Pan Chuxi, Williams David E, Moraes Trevor, Wen Xiao-Yan, Rotstein Ori, Andersen Raymond J, Lee Warren L

Highly oxygenated cyclohexenes from the leaves of Uvaria grandiflora Roxb. ex Hornem and their cytotoxic and α-glucosidase inhibitory activities

从大花乌瓦利亚(Uvaria grandiflora Roxb. ex Hornem)叶片中分离得到的高氧化环己烯及其细胞毒性和α-葡萄糖苷酶抑制活性

Suthiphasilp, Virayu; Betangah, Moses Egoh; Teerapongpisan, Passakorn; Rujanapun, Narawadee; Chaiyosang, Boonyanoot; Tontapha, Sarawut; Kumboonma, Pakit; Patrick, Brian O; Andersen, Raymond J; Charoensup, Rawiwan; Duangyod, Thidarat; Promnart, Phunrawie; Maneerat, Tharakorn; Laphookhieo, Surat

Ex vivo and in vivo HIV-1 latency reversal by "Mukungulu," a protein kinase C-activating African medicinal plant extract

非洲药用植物提取物“Mukungulu”可激活蛋白激酶C,并能逆转体外和体内HIV-1潜伏感染。

Richard, Khumoekae; Yuan, Zhe; Tang, Hsin-Yao; Goldman, Aaron R; Kuthu, Riza; Raphane, Boingotlo; Register, Emery T; Sharma, Paridhima; Ross, Brian N; Morris, Jessicamarie; Williams, David E; Cheney, Carol; Wu, Guoxin; Mounzer, Karam; Laird, Gregory M; Zuck, Paul; Andersen, Raymond J; Simonambango, Sundana; Andrae-Marobela, Kerstin; Tietjen, Ian; Montaner, Luis J

Piperazate-Guided Isolation of Caveamides A and B, Cyclohexenylalanine-Containing Nonribosomal Peptides from a Cave Actinomycete

利用哌拉唑酯导向法从洞穴放线菌中分离出含环己烯基丙氨酸的非核糖体肽——洞穴酰胺A和B

Hagar, Mostafa; Morgan, Kalindi D; Stumpf, Spencer D; Tsingos, Maya; Banuelos, Carmen A; Sadar, Marianne D; Blodgett, Joshua A V; Andersen, Raymond J; Ryan, Katherine S

Synthesis and in vitro assessment of gold nanoparticles conjugated with extracts, sterols and pure compounds derived from marine sponges from the Indian and Pacific Oceans

合成及体外评价源自印度洋和太平洋海洋海绵的提取物、甾醇和纯化合物与金纳米粒子的结合物

Ramanjooloo, Avin; Bekah, Devesh; Adeyemi, Samson A; Ubanako, Philemon; Ngema, Lindokuhle; Choonara, Yahya E; Williams, David E; Polishchuk, Elena A; Andersen, Raymond J; Bhaw-Luximon, Archana

Curcuphenol possesses an unusual histone deacetylase enhancing activity that counters immune escape in metastatic tumours

姜黄酚具有一种不寻常的组蛋白去乙酰化酶增强活性,可对抗转移性肿瘤的免疫逃逸。

Ellis, Samantha L S; Dada, Sarah; Nohara, Lilian L; Saranchova, Iryna; Munro, Lonna; Pfeifer, Cheryl G; Eyford, Brett A; Morova, Tunc; Williams, David E; Cheng, Ping; Lack, Nathan A; Andersen, Raymond J; Jefferies, Wilfred A