Modulating the Binding Kinetics of Bruton's Tyrosine Kinase Inhibitors through Transition-State Effects
通过过渡态效应调节布鲁顿酪氨酸激酶抑制剂的结合动力学
期刊:Journal of the American Chemical Society
影响因子:15.6
doi:10.1021/jacs.5c07063
Bravo, Eduardo Jr; Li, Yong; Lin, David Yin-Wei; Srinivasan, Bharath; Barone, Marco; Li, Stan Xiaogang; DelloRusso, Francesca; Rahiyanath, Anza Suneer; Corrionero, Ana; Alfonso, Patricia; Prendiville, Niall; Kozakov, Dima; Andreotti, Amy H; Tonge, Peter J