日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Safety and efficacy of HSP90 inhibitor ganetespib for neoadjuvant treatment of stage II/III breast cancer

HSP90 抑制剂 Ganetespib 用于 II/III 期乳腺癌新辅助治疗的安全性和有效性

Julie E Lang, Andres Forero-Torres, Douglas Yee, Christina Yau, Denise Wolf, John Park, Barbara A Parker, A Jo Chien, Anne M Wallace, Rashmi Murthy, Kathy S Albain, Erin D Ellis, Heather Beckwith, Barbara B Haley, Anthony D Elias, Judy C Boughey, Rachel L Yung, Claudine Isaacs, Amy S Clark, Hyo S Ha

Preclinical Activity of HER2-Selective Tyrosine Kinase Inhibitor Tucatinib as a Single Agent or in Combination with Trastuzumab or Docetaxel in Solid Tumor Models

HER2 选择性酪氨酸激酶抑制剂 Tucatinib 作为单一药物或与曲妥珠单抗或多西他赛联合用于实体肿瘤模型的临床前活性

Anita Kulukian, Patrice Lee, Janelle Taylor, Robert Rosler, Peter de Vries, Daniel Watson, Andres Forero-Torres, Scott Peterson

O-GlcNAcylation of GLI transcription factors in hyperglycemic conditions augments Hedgehog activity

高血糖条件下 GLI 转录因子的 O-GlcNAc 糖基化增强了 Hedgehog 活性

Shamik Das, Sarah K Bailey, Brandon J Metge, Ann Hanna, Dominique C Hinshaw, Mateus Mota, Andres Forero-Torres, John C Chatham, Rajeev S Samant, Lalita A Shevde

The antitumor effects of entinostat in ovarian cancer require adaptive immunity

恩替诺特在卵巢癌中的抗肿瘤作用需要适应性免疫。

Haller J Smith ,Tyler R McCaw ,Angelina I Londono ,Ashwini A Katre ,Selene Meza-Perez ,Eddy S Yang ,Andres Forero ,Donald J Buchsbaum ,Troy D Randall ,J Michael Straughn Jr ,Lyse A Norian ,Rebecca C Arend

Trastuzumab-Resistant HER2+ Breast Cancer Cells Retain Sensitivity to Poly (ADP-Ribose) Polymerase (PARP) Inhibition

曲妥珠单抗耐药的HER2+乳腺癌细胞仍对聚(ADP-核糖)聚合酶(PARP)抑制剂敏感

Monica E Wielgos ,Zhuo Zhang # ,Rajani Rajbhandari # ,Tiffiny S Cooper ,Ling Zeng ,Andres Forero ,Francisco J Esteva ,C Kent Osborne ,Rachel Schiff ,Albert F LoBuglio ,Susan E Nozell ,Eddy S Yang

Low PTEN levels and PIK3CA mutations predict resistance to neoadjuvant lapatinib and trastuzumab without chemotherapy in patients with HER2 over-expressing breast cancer

低 PTEN 水平和 PIK3CA 突变可预测 HER2 过度表达乳腺癌患者对新辅助拉帕替尼和曲妥珠单抗(未进行化疗)的耐药性

Mothaffar F Rimawi, Carmine De Angelis, Alejandro Contreras, Fresia Pareja, Felipe C Geyer, Kathleen A Burke, Sabrina Herrera, Tao Wang, Ingrid A Mayer, Andres Forero, Rita Nanda, Matthew P Goetz, Jenny C Chang, Ian E Krop, Antonio C Wolff, Anne C Pavlick, Suzanne A W Fuqua, Carolina Gutierrez, Susa

Selective Targeting of Myeloid-Derived Suppressor Cells in Cancer Patients Using DS-8273a, an Agonistic TRAIL-R2 Antibody

使用 DS-8273a(一种激动剂 TRAIL-R2 抗体)选择性靶向癌症患者中的髓系抑制细胞

George A Dominguez, Thomas Condamine, Sridevi Mony, Ayumi Hashimoto, Fang Wang, Qin Liu, Andres Forero, Johanna Bendell, Robert Witt, Neil Hockstein, Prasanna Kumar, Dmitry I Gabrilovich

A Randomized Phase II Neoadjuvant Study of Cisplatin, Paclitaxel With or Without Everolimus in Patients with Stage II/III Triple-Negative Breast Cancer (TNBC): Responses and Long-term Outcome Correlated with Increased Frequency of DNA Damage Response Gene Mutations, TNBC Subtype, AR Status, and Ki67

一项针对 II/III 期三阴性乳腺癌 (TNBC) 患者进行顺铂、紫杉醇联合或不联合依维莫司治疗的随机 II 期新辅助治疗研究:治疗反应和长期结果与 DNA 损伤反应基因突变频率增加、TNBC 亚型、AR 状态和 Ki67 相关

Bojana Jovanović, Ingrid A Mayer, Erica L Mayer, Vandana G Abramson, Aditya Bardia, Melinda E Sanders, M Gabriela Kuba, Monica V Estrada, J Scott Beeler, Timothy M Shaver, Kimberly C Johnson, Violeta Sanchez, Jennifer M Rosenbluth, Patrick M Dillon, Andres Forero-Torres, Jenny C Chang, Ingrid M Mesz

Serum thymidine kinase 1 activity as a pharmacodynamic marker of cyclin-dependent kinase 4/6 inhibition in patients with early-stage breast cancer receiving neoadjuvant palbociclib

血清胸苷激酶 1 活性作为接受新辅助哌柏西利治疗的早期乳腺癌患者细胞周期蛋白依赖性激酶 4/6 抑制的药效学标志

Nusayba Bagegni, Shana Thomas, Ning Liu, Jingqin Luo, Jeremy Hoog, Donald W Northfelt, Matthew P Goetz, Andres Forero, Mattias Bergqvist, Jakob Karen, Magnus Neumüller, Edward M Suh, Zhanfang Guo, Kiran Vij, Souzan Sanati, Matthew Ellis, Cynthia X Ma

Epigenetic modifiers upregulate MHC II and impede ovarian cancer tumor growth

表观遗传修饰因子上调 MHC II 并阻碍卵巢癌肿瘤生长

Taylor B Turner, Selene Meza-Perez, Angelina Londoño, Ashwini Katre, Jacelyn E Peabody, Haller J Smith, Andres Forero, Lyse A Norian, J Michael Straughn Jr, Donald J Buchsbaum, Troy D Randall, Rebecca C Arend