日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cytotoxicity of Zardaverine in Embryonal Rhabdomyosarcoma from a Costello Syndrome Patient

扎达维林对科斯特洛综合征患者胚胎横纹肌肉瘤的细胞毒性

Donna M Cartledge, Katherine M Robbins, Katherine M Drake, Rachel Sternberg, Deborah L Stabley, Karen W Gripp, E Anders Kolb, Katia Sol-Church, Andrew D Napper

A sensitive luminescent assay for the histone methyltransferase NSD1 and other SAM-dependent enzymes

针对组蛋白甲基转移酶 NSD1 和其他 SAM 依赖性酶的灵敏发光检测

Katherine M Drake, Venita G Watson, Anne Kisielewski, Rebecca Glynn, Andrew D Napper

Development of a high-throughput screening-compatible assay for the discovery of inhibitors of the AF4-AF9 interaction using AlphaScreen technology

使用 AlphaScreen 技术开发高通量筛选兼容检测方法,以发现 AF4-AF9 相互作用的抑制剂

Venita Gresham Watson, Katherine M Drake, Yu Peng, Andrew D Napper

Identification of specific inhibitors of human RAD51 recombinase using high-throughput screening

利用高通量筛选鉴定人类 RAD51 重组酶的特异性抑制剂

Fei Huang, Nuzhat A Motlekar, Chelsea M Burgwin, Andrew D Napper, Scott L Diamond, Alexander V Mazin

Parallel High-Throughput Automated Assays to Measure Cell Growth and Beta-Galactosidase Reporter Gene Expression in the Yeast Saccharomyces cerevisiae

平行高通量自动化检测法测量酿酒酵母中的细胞生长和 β-半乳糖苷酶报告基因表达

Andrew D Napper, Nuzhat Motlekar, Rogerio Alves de Almeida, Graham D Pavitt

Identification of triazinoindol-benzimidazolones as nanomolar inhibitors of the Mycobacterium tuberculosis enzyme TDP-6-deoxy-d-xylo-4-hexopyranosid-4-ulose 3,5-epimerase (RmlC)

鉴定三嗪吲哚-苯并咪唑酮为结核分枝杆菌酶 TDP-6-脱氧-d-木糖-4-己吡喃糖苷-4-酮糖 3,5-差向异构酶 (RmlC) 的纳摩尔抑制剂

Sharmila Sivendran, Victoria Jones, Dianqing Sun, Yi Wang, Anna E Grzegorzewicz, Michael S Scherman, Andrew D Napper, J Andrew McCammon, Richard E Lee, Scott L Diamond, Michael McNeil

Discovery of chemical modulators of a conserved translational control pathway by parallel screening in yeast

通过酵母平行筛选发现保守翻译控制途径的化学调节剂

Nuzhat Motlekar, Rogerio Alves de Almeida, Graham D Pavitt, Scott L Diamond, Andrew D Napper

Kinetic characterization and molecular docking of a novel, potent, and selective slow-binding inhibitor of human cathepsin L

新型、强效、选择性慢速结合人类组织蛋白酶 L 抑制剂的动力学表征和分子对接

Parag P Shah, Michael C Myers, Mary Pat Beavers, Jeremy E Purvis, Huiyan Jing, Heather J Grieser, Elizabeth R Sharlow, Andrew D Napper, Donna M Huryn, Barry S Cooperman, Amos B Smith 3rd, Scott L Diamond