日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of 5-(Aryl)amino-1,2,3-triazole-containing 2,1,3-Benzothiadiazoles via Azide-Nitrile Cycloaddition Followed by Buchwald-Hartwig Reaction

通过叠氮化物-腈环加成反应和 Buchwald-Hartwig 反应合成含 5-(芳基)氨基-1,2,3-三唑的 2,1,3-苯并噻二唑

Pavel S Gribanov, Anna N Philippova, Maxim A Topchiy, Dmitry A Lypenko, Artem V Dmitriev, Sergey D Tokarev, Alexander F Smol'yakov, Alexey N Rodionov, Andrey F Asachenko, Sergey N Osipov

New Allosteric Modulators of AMPA Receptors: Synthesis and Study of Their Functional Activity by Radioligand-Receptor Binding Analysis

AMPA 受体的新型变构调节剂:合成并通过放射性配体-受体结合分析研究其功能活性

Elena A Golubeva, Mstislav I Lavrov, Polina N Veremeeva, Tatiana V Vyunova, Konstantin V Shevchenko, Maxim A Topchiy, Andrey F Asachenko, Vladimir A Palyulin

General Method of Synthesis of 5-(Het)arylamino-1,2,3-triazoles via Buchwald-Hartwig Reaction of 5-Amino- or 5-Halo-1,2,3-triazoles

通过 5-氨基或 5-卤代-1,2,3-三唑的 Buchwald-Hartwig 反应合成 5-(杂)芳氨基-1,2,3-三唑的通用方法

Pavel S Gribanov, Anna N Philippova, Maxim A Topchiy, Lidiya I Minaeva, Andrey F Asachenko, Sergey N Osipov

Structure-Activity Relationships and Transcriptomic Analysis of Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitors

缺氧诱导因子脯氨酰羟化酶抑制剂的构效关系及转录组分析

Andrey A Poloznikov, Sergey V Nikulin, Dmitry M Hushpulian, Anna Yu Khristichenko, Andrey I Osipyants, Andrey F Asachenko, Olga V Shurupova, Svyatoslav S Savin, Sue H Lee, Irina N Gaisina, Gregory R J Thatcher, Anthony Narciso, Eric P Chang, Sergey V Kazakov, Nancy Krucher, Vladimir I Tishkov, Bobby