日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In Silico Studies and Biological Evaluation of Thiosemicarbazones as Cruzain-Targeting Trypanocidal Agents for Chagas Disease

利用计算机模拟研究和生物学评价硫代氨基脲类化合物作为靶向克鲁赞锥虫的锥虫杀灭剂治疗恰加斯病

Meier, Lidiane; de Melo, Milena F C V; Abreu, Heitor R; Oliveira, Isabella M E; Sens, Larissa; Doring, Thiago H; Krogh, Renata; Beatriz, Adilson; Andricopulo, Adriano D; Saba, Sumbal; de Oliveira, Aldo S; Rafique, Jamal

Discovery and Early Optimization of 1H-Indole-2-carboxamides with Anti-Trypanosoma cruzi Activity

发现并早期优化具有抗克氏锥虫活性的1H-吲哚-2-甲酰胺类化合物

de Oliveira, Ramon G; Cruz, Luiza R; Dessoy, Marco A; Koovits, Paul J; Dos Santos, Deborah A; de Oliveira, Luiz F N; Ferreira, Rafael A; Mollo, María C; Lee, Eun; Duarte, Simone M; Krogh, Renata; Ferreira, Leonardo L G; Chelucci, Rafael C; Dichiara, Maria; Simpson, Quillon J; Feltrin, Clarissa; da Silva, Adriana C; Dos Santos, Benedito M; Broering, Milena F; Pollastri, Michael P; Ferrins, Lori; Moraes, Carolina B; Andricopulo, Adriano D; Kratz, Jadel M; Sjö, Peter; Mowbray, Charles E; Dias, Luiz C

Design, Synthesis, and In Vitro Evaluation of 4-(Arylchalcogenyl)methyl)-1H-1,2,3-triazol-1-yl-menadione: Exploring Their Potential Against Tuberculosis

4-(芳基硫代基)甲基)-1H-1,2,3-三唑-1-基-甲萘醌的设计、合成及体外评价:探索其抗结核病的潜力

Santos, Nathália L B; Gomes, Luana S; Ribeiro, Ruan C B; Carvalho, Alcione S de; Lourenço, Maria Cristina S; Marins, Laís Machado; Valle, Sandy Polycarpo; Doring, Thiago H; Andricopulo, Adriano D; Oliveira, Aldo S de; Ferreira, Vitor F; da Silva, Fernando de C; Forezi, Luana da Silva Magalhães; Nascimento, Vanessa

Phenotypic Screening of H(1)-Antihistamines Identifies Promethazine and Rupatadine as Active Compounds Against Toxocara canis Infective Larvae

表型筛选H(1)抗组胺药,发现异丙嗪和卢帕他定对犬弓蛔虫感染性幼虫具有活性

Silva, Taís C; Godoy-Silva, Julia; Amaro, Monique C; Silva-Silva, João V; Doring, Thiago H; Ferreira, Leonardo L G; Andricopulo, Adriano D; de Moraes, Josué

In Vitro and In Vivo Evaluation of the Antischistosomal Activity of Polygodial and 9-Deoxymuzigadial Isolated from Drimys brasiliensis Branches

从巴西毛鼠耳蝠枝条中分离得到的聚角醛和9-脱氧穆齐加醛的抗血吸虫活性的体外和体内评价

Umehara, Eric; Cajas, Rayssa A; Conceição, Gabriel B; Antar, Guilherme M; Andricopulo, Adriano D; Moraes, Josué de; Lago, João Henrique G

Hit-to-Lead Studies of Pyrazinylpiperazines against Visceral Leishmaniasis: Pharmacokinetic Profile and In Vivo Efficacy of Potent Compounds against Leishmania infantum.

吡嗪基哌嗪类化合物对内脏利什曼病的先导化合物研究:强效化合物对婴儿利什曼原虫的药代动力学特征和体内疗效

Jacques Dit Lapierre Thibault Joseph William, Gabriela Faleiro de Moura Lodi Cruz Mariza, Barbosa Gisele, Costa Analu R, Chávez-Fumagalli Miguel Angel, Froes Thamires Quadros, Ramos Priscila Zonzini, Macruz Paula Derksen, Carolyne Souza Trindade Thalita, Pilau Eduardo Jorge, Sampaio Tavares Veras Patricia, Nonato Maria Cristina, Massirer Katlin B, Ferreira Leonardo L G, Andricopulo Adriano D, Lima Lídia Moreira, Murta Silvane Maria Fonseca, Rezende Júnior Celso de Oliveira

Latin American Natural Product Database (LANaPDB): An Update

拉丁美洲天然产物数据库(LANaPDB):最新进展

Gómez-García, Alejandro; Acuña Jiménez, Daniel A; Zamora, William J; Barazorda-Ccahuana, Haruna L; Chávez-Fumagalli, Miguel Á; Valli, Marilia; Andricopulo, Adriano D; Bolzani, Vanderlan da S; Olmedo, Dionisio A; Solís, Pablo N; Núñez, Marvin J; Rodríguez Pérez, Johny R; Valencia Sánchez, Hoover A; Cortés Hernández, Héctor F; Mosquera Martinez, Oscar M; Medina-Franco, José L

Neglected Tropical Diseases: A Chemoinformatics Approach for the Use of Biodiversity in Anti-Trypanosomatid Drug Discovery

被忽视的热带病:利用生物多样性进行抗锥虫药物发现的化学信息学方法

Valli, Marilia; Döring, Thiago H; Marx, Edgard; Ferreira, Leonardo L G; Medina-Franco, José L; Andricopulo, Adriano D

Synthesis and Anti-Trypanosoma cruzi Activity of 3-Cyanopyridine Derivatives

3-氰基吡啶衍生物的合成及其抗克氏锥虫活性

Slafer, Brian W; Dessoy, Marco A; de Oliveira, Ramon G; Mollo, Maria C; Lee, Eun; Matheeussen, An; Maes, Louis; Caljon, Guy; Ferreira, Leonardo L G; Krogh, Renata; Andricopulo, Adriano D; Cruz, Luiza R; Mowbray, Charles E; Kratz, Jadel M; Dias, Luiz C

The 3D pharmacophore modeling to explore new antischistosomal agents among US FDA approved drugs

利用三维药效团模型探索美国FDA批准药物中的新型抗血吸虫药物

Dobrachinski, Leandro; Ferreira, Leonardo Lg; Cirino, Maria E; Andrade-de-Siqueira, Allan I; Mafud, Ana C; Mascarenhas, Yvonne P; Andricopulo, Adriano D; de Moraes, Josué