日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Probing the binding of interleukin-23 to individual receptor components and the IL-23 heteromeric receptor complex in living cells using NanoBRET

利用NanoBRET技术探测活细胞中白细胞介素-23与单个受体组分以及IL-23异源受体复合物的结合情况。

Charles S Lay ,Angela Bridges ,Joelle Goulding ,Stephen J Briddon ,Zoja Soloviev ,Peter D Craggs ,Stephen J Hill

Discovery of functionally distinct anti-C7 monoclonal antibodies and stratification of anti-nicotinic AChR positive Myasthenia Gravis patients

发现功能不同的抗 C7 单克隆抗体并对抗烟碱 AChR 阳性重症肌无力患者进行分层

Eleonora Lekova, Wioleta M Zelek, David Gower, Claus Spitzfaden, Isabelle H Osuch, Elen John-Morris, Lasse Stach, Darren Gormley, Andrew Sanderson, Angela Bridges, Elizabeth R Wear, Sebastien Petit-Frere, Michael N Burden, Richard Priest, Trevor Wattam, Semra J Kitchen, Maria Feeney, Susannah Davis,

GSK137, a potent small-molecule BCL6 inhibitor with in vivo activity, suppresses antibody responses in mice

GSK137 是一种具有体内活性的强效小分子 BCL6 抑制剂,可抑制小鼠的抗体反应

Andrew C Pearce, Mark J Bamford, Ruth Barber, Angela Bridges, Maire A Convery, Constantinos Demetriou, Sian Evans, Thomas Gobbetti, David J Hirst, Duncan S Holmes, Jonathan P Hutchinson, Sandrine Jayne, Larissa Lezina, Michael T McCabe, Cassie Messenger, Joanne Morley, Melissa C Musso, Paul Scott-St

Discovery of GSK2795039, a Novel Small Molecule NADPH Oxidase 2 Inhibitor

发现新型小分子 NADPH 氧化酶 2 抑制剂 GSK2795039

Kazufumi Hirano, Woei Shin Chen, Adeline L W Chueng, Angela A Dunne, Tamara Seredenina, Aleksandra Filippova, Sumitra Ramachandran, Angela Bridges, Laiq Chaudry, Gary Pettman, Craig Allan, Sarah Duncan, Kiew Ching Lee, Jean Lim, May Thu Ma, Agnes B Ong, Nicole Y Ye, Shabina Nasir, Sri Mulyanidewi, C

Crystallizing Membrane Proteins in the Lipidic Mesophase. Experience with Human Prostaglandin E2 Synthase 1 and an Evolving Strategy

脂质中间相中的膜蛋白结晶。人类前列腺素 E2 合酶 1 的经验和不断发展的策略

Dianfan Li, Nicole Howe, Abhiram Dukkipati, Syed T A Shah, Benjamin D Bax, Colin Edge, Angela Bridges, Phil Hardwicke, Onkar M P Singh, Ged Giblin, Alexander Pautsch, Roland Pfau, Gisela Schnapp, Meitian Wang, Vincent Olieric, Martin Caffrey

A selective jumonji H3K27 demethylase inhibitor modulates the proinflammatory macrophage response

选择性 jumonji H3K27 去甲基化酶抑制剂调节促炎性巨噬细胞反应

Laurens Kruidenier, Chun-wa Chung, Zhongjun Cheng, John Liddle, KaHing Che, Gerard Joberty, Marcus Bantscheff, Chas Bountra, Angela Bridges, Hawa Diallo, Dirk Eberhard, Sue Hutchinson, Emma Jones, Roy Katso, Melanie Leveridge, Palwinder K Mander, Julie Mosley, Cesar Ramirez-Molina, Paul Rowland, Chr

Over expression of wild type or a catalytically dead mutant of Sirtuin 6 does not influence NFκB responses

野生型或催化失活突变型 Sirtuin 6 的过度表达不会影响 NFκB 反应

Rachel Grimley, Oxana Polyakova, Jessica Vamathevan, Joanne McKenary, Brian Hayes, Champa Patel, Janet Smith, Angela Bridges, Andrew Fosberry, Anshu Bhardwaja, Bernadette Mouzon, Chun-Wa Chung, Nathalie Barrett, Nicola Richmond, Sundip Modha, Roberto Solari

Configuration of a high-content imaging platform for hit identification and pharmacological assessment of JMJD3 demethylase enzyme inhibitors

配置高内涵成像平台用于 JMJD3 去甲基化酶抑制剂的鉴定和药理学评价

Alpa Mulji, Carl Haslam, Fiona Brown, Rebecca Randle, Bhumika Karamshi, Julia Smith, Robert Eagle, Jordi Munoz-Muriedas, Joanna Taylor, Arshad Sheikh, Angela Bridges, Kirsty Gill, Rob Jepras, Penny Smee, Mike Barker, Mike Woodrow, John Liddle, Pamela Thomas, Emma Jones, Laurie Gordon, Rob Tanner, Me