日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Deep-Learning Driven Identification of Novel Antimicrobial Peptides

基于深度学习的新型抗菌肽鉴定

Arino, Silvia; Sgueglia, Gianmattia; Leone, Linda; Oliva, Rosario; Vecchio, Pompea Del; Larrouy-Maumus, Gerald; Lombardi, Angela; De Simone, Alfonso; Nastri, Flavia

Stepwise Structural Simplification of the Dihydroxyanthraquinone Moiety of a Multitarget Rhein-Based Anti-Alzheimer Lead to Improve Drug Metabolism and Pharmacokinetic Properties

逐步简化多靶点大黄酸类抗阿尔茨海默症药物二羟基蒽醌部分的结构以改善药物代谢和药代动力学特性

Caterina Pont, Anna Sampietro, F Javier Pérez-Areales, Nunzia Cristiano, Agustí Albalat, Belén Pérez, Manuela Bartolini, Angela De Simone, Vincenza Andrisano, Marta Barenys, Elisabet Teixidó, Raimon Sabaté, M Isabel Loza, José Brea, Diego Muñoz-Torrero

Integrating a quinone substructure into histone deacetylase inhibitors to cope with Alzheimer's disease and cancer

将醌亚结构整合到组蛋白去乙酰化酶抑制剂中以应对阿尔茨海默病和癌症

Melissa Guardigni, Giulia Greco, Eleonora Poeta, Alan Santini, Elisa Tassinari, Christian Bergamini, Chiara Zalambani, Angela De Simone, Vincenza Andrisano, Elisa Uliassi, Barbara Monti, Maria Laura Bolognesi, Carmela Fimognari, Andrea Milelli

Phenolic and Antioxidant Characterization of Fruit By-Products for Their Nutraceuticals and Dietary Supplements Valorization under a Circular Bio-Economy Approach

循环生物经济方法下水果副产品的酚类和抗氧化剂特性及其作为营养食品和膳食补充剂的价值评估

Cristina Terenzi, Gabriela Bermudez, Francesca Medri, Lara Davani, Vincenzo Tumiatti, Vincenza Andrisano, Serena Montanari, Angela De Simone

Hit Identification and Functional Validation of Novel Dual Inhibitors of HDAC8 and Tubulin Identified by Combining Docking and Molecular Dynamics Simulations

通过结合对接和分子动力学模拟鉴定出 HDAC8 和微管蛋白的新型双重抑制剂的命中鉴定和功能验证

Antonio Curcio, Roberta Rocca, Federica Chiera, Maria Eugenia Gallo Cantafio, Ilenia Valentino, Ludovica Ganino, Pierpaolo Murfone, Angela De Simone, Giulia Di Napoli, Stefano Alcaro, Nicola Amodio, Anna Artese

Quantum Mechanical Predictions of the Antioxidant Capability of Moracin C Isomers

莫拉辛C异构体抗氧化能力的量子力学预测

Parise, Angela; De Simone, Bruna Clara; Marino, Tiziana; Toscano, Marirosa; Russo, Nino

Derivatives of the β-Crinane Amaryllidaceae Alkaloid Haemanthamine as Multi-Target Directed Ligands for Alzheimer's Disease

β-克里烷石蒜科生物碱海金花胺衍生物作为阿尔茨海默病的多靶点定向配体

Eliška Kohelová, Rozálie Peřinová, Negar Maafi, Jan Korábečný, Daniela Hulcová, Jana Maříková, Tomáš Kučera, Loreto Martínez González, Martina Hrabinova, Katarina Vorčáková, Lucie Nováková, Angela De Simone, Radim Havelek, Lucie Cahlíková6

Investigating in Vitro Amyloid Peptide 1-42 Aggregation: Impact of Higher Molecular Weight Stable Adducts

研究体外淀粉样肽 1-42 聚集:高分子量稳定加合物的影响

Angela De Simone, Marina Naldi, Daniele Tedesco, Andrea Milelli, Manuela Bartolini, Lara Davani, Darius Widera, Mark L Dallas, Vincenza Andrisano

Amaryllidaceae Alkaloids as Potential Glycogen Synthase Kinase-3β Inhibitors

石蒜科生物碱作为潜在的糖原合酶激酶-3β 抑制剂

Daniela Hulcová, Kateřina Breiterová, Tomáš Siatka, Kamila Klímová, Lara Davani, Marcela Šafratová, Anna Hošťálková, Angela De Simone, Vincenza Andrisano, Lucie Cahlíková1