日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of Stereoenriched Piperidines via Chemo-Enzymatic Dearomatization of Activated Pyridines

通过活化吡啶的化学酶法脱芳构化合成立体富集的哌啶

Harawa, Vanessa; Thorpe, Thomas W; Marshall, James R; Sangster, Jack J; Gilio, Amelia K; Pirvu, Lucian; Heath, Rachel S; Angelastro, Antonio; Finnigan, James D; Charnock, Simon J; Nafie, Jordan W; Grogan, Gideon; Whitehead, Roger C; Turner, Nicholas J

Galactose Oxidase Enables Modular Assembly of Conjugates from Native Antibodies with High Drug-to-Antibody Ratios

半乳糖氧化酶能够以高药物抗体比,从天然抗体出发,模块化组装偶联物

Angelastro, Antonio; Barkhanskiy, Alexey; Mattey, Ashley P; Pallister, Edward G; Spiess, Reynard; Goundry, William; Barran, Perdita; Flitsch, Sabine L

Loss of Hyperconjugative Effects Drives Hydride Transfer during Dihydrofolate Reductase Catalysis.

超共轭效应的丧失驱动二氢叶酸还原酶催化过程中的氢化物转移

Angelastro Antonio, Ruiz-Pernía J Javier, Tuñón Iñaki, Moliner Vicent, Luk Louis Y P, Allemann Rudolf K

Reactivity and Selectivity of Iminium Organocatalysis Improved by a Protein Host

蛋白质宿主可提高亚胺有机催化的反应活性和选择性

Nödling, Alexander R; Świderek, Katarzyna; Castillo, Raquel; Hall, Jonathan W; Angelastro, Antonio; Morrill, Louis C; Jin, Yi; Tsai, Yu-Hsuan; Moliner, Vicent; Luk, Louis Y P