A covalent fragment-based strategy targeting a novel cysteine to inhibit activity of mutant EGFR kinase
一种基于共价片段的策略，靶向一种新型半胱氨酸，以抑制突变型EGFR激酶的活性。
期刊:RSC Medicinal Chemistry
影响因子:3.6
doi:10.1039/d3md00439b
Kuki, Naoki; Walmsley, David L; Kanai, Kazuo; Takechi, Sho; Yoshida, Masao; Murakami, Ryo; Takano, Kohei; Tominaga, Yuichi; Takahashi, Mizuki; Ito, Shuichiro; Nakao, Naoki; Angove, Hayley; Baker, Lisa M; Carter, Edward; Dokurno, Pawel; Le Strat, Loic; Macias, Alba T; Molyneaux, Carrie-Anne; Murray, James B; Surgenor, Allan E; Hamada, Tomoaki; Hubbard, Roderick E
