Expanding the knowledge around antitubercular 5-(2-aminothiazol-4-yl)isoxazole-3-carboxamides: Hit-to-lead optimization and release of a novel antitubercular chemotype via scaffold derivatization
扩展有关抗结核药物 5-(2-氨基噻唑-4-基)异恶唑-3-甲酰胺的认识:通过支架衍生化进行先导化合物优化和新型抗结核化学型的释放
期刊:European Journal of Medicinal Chemistry
影响因子:6
doi:10.1016/j.ejmech.2022.114916
Miriam Girardini, Francesca Ferlenghi, Giannamaria Annunziato, Giulia Degiacomi, Bianca Papotti, Cinzia Marchi, José Camilla Sammartino, Sari S Rasheed, Anna Contini, Maria Rosalia Pasca, Federica Vacondio, Joanna C Evans, Thomas Dick, Rolf Müller, Gabriele Costantino, Marco Pieroni