日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacokinetics, safety, and tolerability of inhaled remdesivir in healthy participants

吸入瑞德西韦在健康受试者中的药代动力学、安全性和耐受性

Humeniuk, Rita; Juneja, Kavita; Chen, Shuguang; Ellis, Scott; Anoshchenko, Olena; Xiao, Deqing; Share, Aaron; Johnston, Matthew; Davies, Santosh; DeZure, Adam; Llewellyn, Joe; Osinusi, Anu; Winter, Helen; Girish, Sandhya; Palaparthy, Ramesh; Dresser, Mark

Characterizing and Quantifying Extrahepatic Metabolism of (-)-Δ9-Tetrahydrocannabinol (THC) and Its Psychoactive Metabolite, (±)-11-Hydroxy-Δ9-THC (11-OH-THC)

表征和量化 (-)-Δ9-四氢大麻酚 (THC) 及其精神活性代谢物 (±)-11-羟基-Δ9-THC (11-OH-THC) 的肝外代谢

Aditya R Kumar, Gabriela I Patilea-Vrana, Olena Anoshchenko, Jashvant D Unadkat

Successful Prediction of Human Steady-State Unbound Brain-to-Plasma Concentration Ratio of P-gp Substrates Using the Proteomics-Informed Relative Expression Factor Approach

利用蛋白质组学指导的相对表达因子方法成功预测人脑血浆中P-gp底物的稳态游离浓度比

Storelli, Flavia; Anoshchenko, Olena; Unadkat, Jashvant D

Novel Trifluoromethyl Pyrimidinone Compounds With Activity Against Mycobacterium tuberculosis

新型三氟甲基嘧啶酮化合物对结核分枝杆菌具有活性

Hembre, Erik; Early, Julie V; Odingo, Joshua; Shelton, Catherine; Anoshchenko, Olena; Guzman, Junitta; Flint, Lindsay; Dennison, Devon; McNeil, Matthew B; Korkegian, Aaron; Ovechkina, Yulia; Ornstein, Paul; Masquelin, Thierry; Hipskind, Philip A; Parish, Tanya

Successful Prediction of Human Fetal Exposure to P-Glycoprotein Substrate Drugs Using the Proteomics-Informed Relative Expression Factor Approach and PBPK Modeling and Simulation

利用蛋白质组学指导的相对表达因子方法和生理药代动力学建模与模拟成功预测人类胎儿对P-糖蛋白底物药物的暴露情况

Anoshchenko, Olena; Storelli, Flavia; Unadkat, Jashvant D

Estimating fetal exposure to the P-gp substrates, corticosteroids, by PBPK modeling to inform prevention of neonatal respiratory distress syndrome

利用生理药代动力学模型估算胎儿对P-gp底物(皮质类固醇)的暴露量,以指导新生儿呼吸窘迫综合征的预防。

Anoshchenko, Olena; Milad, Mark A; Unadkat, Jashvant D

Gestational Age-Dependent Abundance of Human Placental Transporters as Determined by Quantitative Targeted Proteomics

通过定量靶向蛋白质组学测定人胎盘转运蛋白的丰度与妊娠年龄的关系

Anoshchenko, Olena; Prasad, Bhagwat; Neradugomma, Naveen K; Wang, Joanne; Mao, Qingcheng; Unadkat, Jashvant D

Hepatic Enzymes Relevant to the Disposition of (-)-∆(9)-Tetrahydrocannabinol (THC) and Its Psychoactive Metabolite, 11-OH-THC

与 (-)-Δ(9)-四氢大麻酚 (THC) 及其精神活性代谢物 11-OH-THC 的处置相关的肝酶

Patilea-Vrana, Gabriela I; Anoshchenko, Olena; Unadkat, Jashvant D