日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.

吗啡烷衍生的双重μ-κ阿片受体激动剂镇痛药的合成与药理学研究

Varga Balazs R, Uprety Rajendra, Paul Barnali, Knoll Alexis, Ramos-Gonzalez Nokomis, Appourchaux Kevin, Taylor Tori, Turgutalp Bengisu, Shinouchi Ryosuke, Eans Shainnel O, Williams Ashai K, Vasquez-Grinnell Steven G, Zaidi Saheem, Nazarova Antonina L, Varadi Andras, Le Rouzic Valerie, Brown Taylor G, Martinez Shani, Ansonoff Michael, Dardashti Rebecca Notis, Hunkele Amanda, Subrath Joan, Welch Matthew, Xu Jin, Rossi Grace C, Pintar John, Pasternak Gavril W, Katritch Vsevolod, McLaughlin Jay P, Pan Ying Xian, Majumdar Susruta

7-Hydroxymitragynine Is an Active Metabolite of Mitragynine and a Key Mediator of Its Analgesic Effects

7-羟基帽柱木碱是帽柱木碱的活性代谢产物,也是其镇痛作用的关键介质。

Kruegel, Andrew C; Uprety, Rajendra; Grinnell, Steven G; Langreck, Cory; Pekarskaya, Elizabeth A; Le Rouzic, Valerie; Ansonoff, Michael; Gassaway, Madalee M; Pintar, John E; Pasternak, Gavril W; Javitch, Jonathan A; Majumdar, Susruta; Sames, Dalibor

Opioids and opioid receptors orchestrate wound repair

阿片类物质和阿片受体协调伤口修复

Wang, Ying; Gupta, Mihir; Poonawala, Tasneem; Farooqui, Mariya; Li, Yunfang; Peng, Fei; Rao, Sheldon; Ansonoff, Michael; Pintar, John E; Gupta, Kalpna

Preclinical findings predicting efficacy and side-effect profile of LY2940094, an antagonist of nociceptin receptors

预测LY2940094(一种伤害感受素受体拮抗剂)疗效和副作用的临床前研究结果

Witkin, Jeffrey M; Rorick-Kehn, Linda M; Benvenga, Mark J; Adams, Benjamin L; Gleason, Scott D; Knitowski, Karen M; Li, Xia; Chaney, Steven; Falcone, Julie F; Smith, Janice W; Foss, Julie; Lloyd, Kirsti; Catlow, John T; McKinzie, David L; Svensson, Kjell A; Barth, Vanessa N; Toledo, Miguel A; Diaz, Nuria; Lafuente, Celia; Jiménez, Alma; Benito, Alfonso; Pedregal, Conception; Martínez-Grau, Maria A; Post, Anke; Ansonoff, Michael A; Pintar, John E; Statnick, Michael A

Mediation of buprenorphine analgesia by a combination of traditional and truncated mu opioid receptor splice variants

丁丙诺啡镇痛作用是通过传统和截短的μ阿片受体剪接变体的组合介导的

Grinnell, Steven G; Ansonoff, Michael; Marrone, Gina F; Lu, Zhigang; Narayan, Ankita; Xu, Jin; Rossi, Grace; Majumdar, Susruta; Pan, Ying-Xian; Bassoni, Daniel L; Pintar, John; Pasternak, Gavril W

The biology of Nociceptin/Orphanin FQ (N/OFQ) related to obesity, stress, anxiety, mood, and drug dependence

伤害感受素/孤啡肽FQ (N/OFQ) 的生物学特性与肥胖、压力、焦虑、情绪和药物依赖有关

Witkin, Jeffrey M; Statnick, Michael A; Rorick-Kehn, Linda M; Pintar, John E; Ansonoff, Michael; Chen, Yanyun; Tucker, R Craig; Ciccocioppo, Roberto

The tail pigmentation pattern of C57BL/6J mice affects nociception/pain quantification in the tail flick test

C57BL/6J小鼠的尾部色素沉着模式会影响甩尾试验中的伤害感受/疼痛量化。

Wen, Ting; Ansonoff, Michael A; Pintar, John E

Codeine and 6-acetylcodeine analgesia in mice

小鼠可待因和6-乙酰可待因镇痛作用

Milo, Steven; Ansonoff, Michael; King, Michael; Rossi, Grace C; Zuckerman, Amy; Pintar, John; Pasternak, Gavril W