日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Chemical Probes Portal - 2024: update on this public resource to support best-practice selection and use of small molecules in biomedical research

化学探针门户网站 - 2024:更新此公共资源,以支持生物医学研究中小分子的最佳实践选择和使用

Sanfelice, Domenico; Antolin, Albert A; Crisp, Alisa; Chen, Yi; Bellenie, Benjamin; Brennan, Paul E; Edwards, Aled; Müller, Susanne; Al-Lazikani, Bissan; Workman, Paul

Concurrence of FGFR1 mutations modulates oncogenesis in glioneuronal tumors.

FGFR1 突变的并发会调节神经胶质肿瘤的发生。

Boni Jacopo, Fernández-González Míriam, Han HyeRim, Roca Carla, Wong Cassandra J, Rioja Cristina, Nogué Clara, Manen-Freixa Leticia, Boulais Jonathan, Torres-Urtizberea Endika, Gomez Antonio, Hasselblatt Martin, Estrada-Tejedor Roger, Antolin Albert A, Elkholi Islam E, Jabado Nada, Côté Jean-François, Gingras Anne-Claude, Rivera Barbara

Elucidating Compound Mechanism of Action and Polypharmacology with a Large-scale Perturbational Profile Compendium

利用大规模扰动谱汇编阐明化合物的作用机制和多药理学

Hu, Lucas ZhongMing; Hirschhorn, Tal; Douglass, Eugene; Murray, Diana; Trudeau, Stephen J; Turunen, Mikko; Pampou, Sergey; Grunn, Adina; Realubit, Ron; Antolin, Albert A; Wang, Alexander L E; Li, Hai; Subramaniam, Prem; Mundi, Prabhjot S; Karan, Charles; Alvarez, Mariano; Honig, Barry; Stockwell, Brent R; Califano, Andrea

Computational repurposing of oncology drugs through off-target drug binding interactions from pharmacological databases

利用药理数据库中非靶向药物结合相互作用进行肿瘤药物的计算再利用

Walpole, Imogen R; Zaman, Farzana Y; Zhao, Peinan; Marshall, Vikki M; Lin, Frank P; Thomas, David M; Shackleton, Mark; Antolin, Albert A; Ameratunga, Malaka

Combining Data-Driven and Structure-Based Approaches in Designing Dual PARP1-BRD4 Inhibitors for Breast Cancer Treatment

结合数据驱动和结构驱动方法设计用于乳腺癌治疗的双重PARP1-BRD4抑制剂

Feng, Bo; Yu, Hui; Dong, Xu; Díaz-Holguín, Alejandro; Antolin, Albert A; Hu, Huabin

canSAR: update to the cancer translational research and drug discovery knowledgebase

canSAR:癌症转化研究和药物发现知识库的更新

di Micco, Patrizio; Antolin, Albert A; Mitsopoulos, Costas; Villasclaras-Fernandez, Eloy; Sanfelice, Domenico; Dolciami, Daniela; Ramagiri, Pradeep; Mica, Ioan L; Tym, Joseph E; Gingrich, Philip W; Hu, Huabin; Workman, Paul; Al-Lazikani, Bissan

The Chemical Probes Portal: an expert review-based public resource to empower chemical probe assessment, selection and use

化学探针门户网站:一个基于专家评审的公共资源,旨在促进化学探针的评估、选择和使用。

Antolin, Albert A; Sanfelice, Domenico; Crisp, Alisa; Villasclaras Fernandez, Eloy; Mica, Ioan L; Chen, Yi; Collins, Ian; Edwards, Aled; Müller, Susanne; Al-Lazikani, Bissan; Workman, Paul

Target 2035 - an update on private sector contributions

2035年目标——私营部门贡献的最新情况

Ackloo, Suzanne; Antolin, Albert A; Bartolome, Jose Manuel; Beck, Hartmut; Bullock, Alex; Betz, Ulrich A K; Böttcher, Jark; Brown, Peter J; Chaturvedi, Menorca; Crisp, Alisa; Daniels, Danette; Dreher, Jan; Edfeldt, Kristina; Edwards, Aled M; Egner, Ursula; Elkins, Jon; Fischer, Christian; Glendorf, Tine; Goldberg, Steven; Hartung, Ingo V; Hillisch, Alexander; Homan, Evert; Knapp, Stefan; Köster, Markus; Krämer, Oliver; Llaveria, Josep; Lessel, Uta; Lindemann, Sven; Linderoth, Lars; Matsui, Hisanori; Michel, Maurice; Montel, Florian; Mueller-Fahrnow, Anke; Müller, Susanne; Owen, Dafydd R; Saikatendu, Kumar Singh; Santhakumar, Vijayaratnam; Sanderson, Wendy; Scholten, Cora; Schapira, Matthieu; Sharma, Sujata; Shireman, Brock; Sundström, Michael; Todd, Matthew H; Tredup, Claudia; Venable, Jennifer; Willson, Timothy M; Arrowsmith, Cheryl H

canSAR chemistry registration and standardization pipeline

canSAR 化学物质注册和标准化流程

Dolciami, Daniela; Villasclaras-Fernandez, Eloy; Kannas, Christos; Meniconi, Mirco; Al-Lazikani, Bissan; Antolin, Albert A

canSAR: update to the cancer translational research and drug discovery knowledgebase

canSAR:癌症转化研究和药物发现知识库的更新

Mitsopoulos, Costas; Di Micco, Patrizio; Fernandez, Eloy Villasclaras; Dolciami, Daniela; Holt, Esty; Mica, Ioan L; Coker, Elizabeth A; Tym, Joseph E; Campbell, James; Che, Ka Hing; Ozer, Bugra; Kannas, Christos; Antolin, Albert A; Workman, Paul; Al-Lazikani, Bissan