Identification of a potent, state-dependent inhibitor of Nav1.7 with oral efficacy in the formalin model of persistent pain
鉴定出一种有效的、状态依赖性的 Nav1.7 抑制剂,在福尔马林持续性疼痛模型中具有口服疗效
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm200018k
Howard Bregman, Loren Berry, John L Buchanan, April Chen, Bingfan Du, Elma Feric, Markus Hierl, Liyue Huang, David Immke, Brett Janosky, Danielle Johnson, Xingwen Li, Joseph Ligutti, Dong Liu, Annika Malmberg, David Matson, Jeff McDermott, Peter Miu, Hanh Nho Nguyen, Vinod F Patel, Daniel Waldon, Be