日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Conformationally Constrained Isoquinolinones as Orally Efficacious Hepatitis B Capsid Assembly Modulators

构象受限的异喹啉酮类化合物作为口服有效的乙型肝炎病毒衣壳组装调节剂

Mesaros, Eugen F; Cole, Andrew G; Kultgen, Steven G; Mani, Nagraj; Fan, Kristi Yi; Dugan, Benjamin J; Ardzinski, Andrzej; Stever, Kim; Micolochick Steuer, Holly M; Graves, Ingrid; Tang, Sunny; Harasym, Troy O; Lam, Angela M; Thi, Emily P; Dorsey, Bruce D; Sofia, Michael J

Preclinical Antiviral and Safety Profiling of the HBV RNA Destabilizer AB-161

乙肝病毒RNA破坏剂AB-161的临床前抗病毒活性和安全性分析

Lam, Angela M; Dugyala, Ravi R; Sheraz, Muhammed; Liu, Fei; Thi, Emily P; Graves, Ingrid E; Cuconati, Andrea; Steuer, Holly Micolochick; Ardzinski, Andrzej; Overholt, Nathan; Mason, Jeremy D; Gotchev, Dimitar; Cole, Andrew G; Harasym, Troy O; Sofia, Michael J

Preclinical Profile of AB-423, an Inhibitor of Hepatitis B Virus Pregenomic RNA Encapsidation

乙肝病毒基因组 RNA 衣壳化抑制剂 AB-423 的临床前概况

Nagraj Mani, Andrew G Cole, Janet R Phelps, Andrzej Ardzinski, Kyle D Cobarrubias, Andrea Cuconati, Bruce D Dorsey, Ellen Evangelista, Kristi Fan, Fang Guo, Haitao Guo, Ju-Tao Guo, Troy O Harasym, Salam Kadhim, Steven G Kultgen, Amy C H Lee, Alice H L Li, Quanxin Long, Sara A Majeski, Richeng Mao, K

Genotypic and phenotypic analyses of hepatitis C virus variants observed in clinical studies of VX-222, a nonnucleoside NS5B polymerase inhibitor

对非核苷类NS5B聚合酶抑制剂VX-222临床研究中观察到的丙型肝炎病毒变异株进行基因型和表型分析

Jiang, Min; Zhang, Eileen Z; Ardzinski, Andrzej; Tigges, Ann; Davis, Andrew; Sullivan, James C; Nelson, Michelle; Spanks, Joan; Dorrian, Jennifer; Nicolas, Olivier; Bartels, Doug J; Rao, B Govinda; Rijnbrand, Rene; Kieffer, Tara L

In vitro phenotypic characterization of hepatitis C virus NS3 protease variants observed in clinical studies of telaprevir

在特拉匹韦临床研究中观察到的丙型肝炎病毒NS3蛋白酶变体的体外表型特征

Jiang, Min; Mani, Nagraj; Lin, Chao; Ardzinski, Andrzej; Nelson, Michelle; Reagan, Dugan; Bartels, Doug; Zhou, Yi; Nicolas, Olivier; Rao, B Govinda; Müh, Ute; Hanzelka, Brian; Tigges, Ann; Rijnbrand, Rene; Kieffer, Tara L