日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Modulation of the 14-3-3σ/C-RAF "Auto"inhibited Complex by Molecular Glues

分子胶对 14-3-3σ/C-RAF“自身”抑制复合物的调节

Konstantinidou, Markella; Vickery, Holly R; Pennings, Marloes A M; Virta, Johanna M; Luo, Shu Yue; Visser, Emira J; Bannier, Sean D; Srikanth, Mrudula; Cismoski, Sabine Z; Young, Lucy C; van den Oetelaar, Maxime C M; McCormick, Frank; Ottmann, Christian; Brunsveld, Luc; Arkin, Michelle R

Stabilization of Native Protein-Protein Interactions with Molecular Glues: A 14-3-3 Case Study

利用分子胶稳定天然蛋白质-蛋白质相互作用:14-3-3 案例研究

Konstantinidou, Markella; Virta, Johanna M; Arkin, Michelle R

Scaffold-hopping for molecular glues targeting the 14-3-3/ERα complex.

针对 14-3-3/ERα 复合物的分子胶的支架跃迁

Konstantinidou Markella, Zingiridis Marios, Pennings Marloes A M, Fragkiadakis Michael, Virta Johanna M, Revalde Jezrael L, Visser Emira J, Ottmann Christian, Brunsveld Luc, Neochoritis Constantinos G, Arkin Michelle R

Opposing role of phagocytic receptors MERTK and AXL in Progranulin deficient FTD.

吞噬受体 MERTK 和 AXL 在前粒蛋白缺乏型 FTD 中的相反作用

Clelland Claire Dudley, Fan Li, Saloner Rowan, Etchegaray Jon Iker, Altobelli Chad Richard, Salomonsson Sally, Maltos Alisha M, Sachdev Aradhana, Zhu Jingjie, Lee Se-In, Li Yaqiao, Zhou Yungui, Le David, Wang Chao, Carling Gillian, Kodama Lay, Sayed Faten, Perez-Bermejo Jaun A, Geier Ethan G, Yokoyama Jennifer S, Rosen Howie, Nana Alissa L, Spina Salvatore, Grinberg Lea T, Seeley William W, Elahi Fanny, Boxer Adam L, Arkin Michelle R, Gan Li

Modulation of the 14-3-3σ/C-RAF "auto"inhibited complex by molecular glues

分子胶对14-3-3σ/C-RAF“自身”抑制复合物的调节

Konstantinidou, Markella; Vickery, Holly R; Pennings, Marloes A M; Virta, Johanna M; Visser, Emira J; Bannier, Sean D; Srikanth, Mrudula; Cismoski, Sabine Z; Young, Lucy C; van den Oetelaar, Maxime C M; McCormick, Frank; Ottmann, Christian; Brunsveld, Luc; Arkin, Michelle R

Deep phenotypic profiling of neuroactive drugs in larval zebrafish

对斑马鱼幼体中神经活性药物进行深度表型分析

Gendelev, Leo; Taylor, Jack; Myers-Turnbull, Douglas; Chen, Steven; McCarroll, Matthew N; Arkin, Michelle R; Kokel, David; Keiser, Michael J

Synthetic autophagy receptor

合成自噬受体

Jiang, Ziwen; Kuo, Yu-Hsuan; Arkin, Michelle R

Synthetic Lethal Targeting of CDK12-Deficient Prostate Cancer with PARP Inhibitors.

利用 PARP 抑制剂对 CDK12 缺陷型前列腺癌进行合成致死靶向治疗

Chou Jonathan, Robinson Troy M, Egusa Emily A, Lodha Roshan, Zhang Meng, Badura Michelle, Mikayelyan Mane, Delavan Henry M, Swinderman Jason, Wilson Chris, Zhu Jun, Das Rajdeep, Nguyen Minh, Loehr Andrea, Golsorkhi Tony, Simmons Andrew, Abida Wassim, Chinnaiyan Arul M, Arkin Michelle R, Small Eric J, Quigley David A, Yang Lixing, Kim Minkyu, Ashworth Alan, Feng Felix Y

Molecular glues for protein-protein interactions: Progressing toward a new dream

用于蛋白质-蛋白质相互作用的分子胶:迈向新的梦想

Konstantinidou, Markella; Arkin, Michelle R

Identifying ligands for the PHD1 finger of KDM5A through high-throughput screening

通过高通量筛选鉴定KDM5A的PHD1指状结构域的配体

Ortiz, Gloria; Longbotham, James E; Qin, Sophia L; Zhang, Meng Yao; Lee, Gregory M; Neitz, R Jeffrey; Kelly, Mark J S; Arkin, Michelle R; Fujimori, Danica Galonić