日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Macrocyclic Myeloid Cell Leukemia 1 (Mcl-1) Inhibitors that Demonstrate Potent Cellular Efficacy and In Vivo Activity in a Mouse Solid Tumor Xenograft Model

发现具有强效细胞活性和在小鼠实体瘤异种移植模型中体内活性的巨环髓系细胞白血病1 (Mcl-1) 抑制剂

Tarr, James C; Jeon, Kyuok; Veerasamy, Nagarathanam; Aichinger, Martin; Salovich, James M; Zhao, Bin; Sensintaffar, John L; Arnhof, Heribert; Wunberg, Tobias; Sgubin, Danielle; Arnold, Allison; Vekariya, Rakesh H; Christov, Plamen P; Kim, Kwangho; Fuchs, Julian Emanuel; Karier, Pol; Betzemeier, Bodo; Van Meveren, Mayme; Miriyala, Nagaraju; Olejniczak, Edward T; Engelhardt, Harald; Lee, Taekyu; McConnell, Darryl; Fesik, Stephen W

Discovery of BI-2493, a Pan-KRAS Inhibitor Showing In Vivo Efficacy.

发现 BI-2493,一种泛 KRAS 抑制剂,显示出体内疗效

Bröker Joachim, Waterson Alex G, Hodges Timothy R, Abbott Jason R, Arnold Allison, Böttcher Jark, Braun Nina, Cui Jianwen, Fuchs Julian E, Gerstberger Thomas, Gogg Sebastian, Hanner Sabine, Herdeis Lorenz, Howell Lucas W, Mantoulidis Andreas, Mayer Moriz, Phan Jason, Rocchetti Francesca, Sankar Kyra, Sarkar Dhruba, Schaaf Otmar, Sensintaffar John L, Sun Qi, Wunberg Tobias, Fesik Stephen W

Differences in Abdominal Muscle Thickness, Strength, and Endurance in Persons Who Are Runners, Active, and Inactive

跑步者、活跃人群和不活跃人群的腹肌厚度、力量和耐力存在差异

Schaeffer, Beth H; Anemaet, Wendy K; Arnold, Allison L; Brabham, Autumn B; Groom, Nancy K; Moore, Cassidee R

Discovery and Structure-Based Optimization of Benzimidazole-Derived Activators of SOS1-Mediated Nucleotide Exchange on RAS

苯并咪唑衍生物激活剂对 RAS 上 SOS1 介导的核苷酸交换的发现和基于结构的优化

Hodges, Timothy R; Abbott, Jason R; Little, Andrew J; Sarkar, Dhruba; Salovich, James M; Howes, Jennifer E; Akan, Denis T; Sai, Jiqing; Arnold, Allison L; Browning, Carrie; Burns, Michael C; Sobolik, Tammy; Sun, Qi; Beesetty, Yugandhar; Coker, Jesse A; Scharn, Dirk; Stadtmueller, Heinz; Rossanese, Olivia W; Phan, Jason; Waterson, Alex G; McConnell, Darryl B; Fesik, Stephen W

Why are Antagonist Muscles Co-activated in My Simulation? A Musculoskeletal Model for Analysing Human Locomotor Tasks

为什么我的模拟中拮抗肌会协同激活?用于分析人类运动任务的肌肉骨骼模型

Lai, Adrian K M; Arnold, Allison S; Wakeling, James M

Quantifying Achilles tendon force in vivo from ultrasound images

利用超声图像量化体内跟腱力

Dick, Taylor J M; Arnold, Allison S; Wakeling, James M

Validation of Hill-type muscle models in relation to neuromuscular recruitment and force-velocity properties: predicting patterns of in vivo muscle force

验证Hill型肌肉模型与神经肌肉募集和力-速度特性的关系:预测体内肌肉力量模式

Biewener, Andrew A; Wakeling, James M; Lee, Sabrina S; Arnold, Allison S

Modulation of joint moments and work in the goat hindlimb with locomotor speed and surface grade

山羊后肢关节力矩和做功随运动速度和路面坡度的变化

Arnold, Allison S; Lee, David V; Biewener, Andrew A

A muscle's force depends on the recruitment patterns of its fibers

肌肉的力量取决于其肌纤维的募集模式。

Wakeling, James M; Lee, Sabrina S M; Arnold, Allison S; de Boef Miara, Maria; Biewener, Andrew A

There is always a trade-off between speed and force in a lever system: comment on McHenry (2010)

在杠杆系统中,速度和力之间总是存在权衡:评论 McHenry (2010)

Arnold, Allison S; Richards, Christopher T; Ros, Ivo G; Biewener, Andrew A