日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

From Concepts to Inhibitors: A Blueprint for Targeting Protein-Protein Interactions

从概念到抑制剂:靶向蛋白质-蛋白质相互作用的蓝图

Hong, Seong Ho; Nguyen, Thu; Ongkingco, Joseph F; Nazzaro, Alex; Arora, Paramjit S

Reengineering of a Proteomimetic Pan-Ras Inhibitor into a Ras Degrader

将一种拟蛋白泛Ras抑制剂改造为Ras降解剂

Ongkingco, Joseph F; Hong, Seong Ho; Toth, Eugene D; Nguyen, Thu; Arora, Paramjit S

Proteomimetic Strategy for the Modulation of Intrinsically Disordered Protein MYC

利用蛋白质模拟策略调控固有无序蛋白MYC

Nguyen, Thu; Hong, Seong Ho; Arora, Paramjit S

Small Molecule Catalyst for Peptide Synthesis

用于肽合成的小分子催化剂

Panigrahi, Nihar R; Khan, Shahrukh M; Handoko; Arora, Paramjit S

C2230, a preferential use- and state-dependent CaV2.2 channel blocker, mitigates pain behaviors across multiple pain models.

C2230 是一种优先使用和状态依赖的 CaV2.2 通道阻滞剂,可减轻多种疼痛模型中的疼痛行为

Tang Cheng, Gomez Kimberly, Chen Yan, Allen Heather N, Hestehave Sara, Rodríguez-Palma Erick J, Loya-Lopez Santiago, Calderon-Rivera Aida, Duran Paz, Nelson Tyler S, Kanumuri Siva Rama Raju, Shah Bijal, Panigrahi Nihar R, Perez-Miller Samantha, Schackmuth Morgan K, Ruparel Shivani, Patwardhan Amol, Price Theodore J, Arora Paramjit S, Sharma Ravindra K, Sharma Abhisheak, Yu Jie, Korczeniewska Olga A, Khanna Rajesh

An Encodable Scaffold for Sequence-Specific Recognition of Duplex RNA

用于双链RNA序列特异性识别的可编码支架

Kwok, Jonathan G; Yuan, Zhi; Arora, Paramjit S

Macrocyclic β-Sheets Stabilized by Hydrogen Bond Surrogates

由氢键替代物稳定的大环β-折叠

Nazzaro, Alex; Lu, Brandon; Sawyer, Nicholas; Watkins, Andrew M; Arora, Paramjit S

A peptidomimetic modulator of the Ca(V)2.2 N-type calcium channel for chronic pain

一种用于治疗慢性疼痛的 Ca(V)2.2 N 型钙通道的肽模拟调节剂

Gomez, Kimberly; Santiago, Ulises; Nelson, Tyler S; Allen, Heather N; Calderon-Rivera, Aida; Hestehave, Sara; Rodríguez Palma, Erick J; Zhou, Yuan; Duran, Paz; Loya-Lopez, Santiago; Zhu, Elaine; Kumar, Upasana; Shields, Rory; Koseli, Eda; McKiver, Bryan; Giuvelis, Denise; Zuo, Wanhong; Inyang, Kufreobong E; Dorame, Angie; Chefdeville, Aude; Ran, Dongzhi; Perez-Miller, Samantha; Lu, Yi; Liu, Xia; Handoko; Arora, Paramjit S; Patek, Marcel; Moutal, Aubin; Khanna, May; Hu, Huijuan; Laumet, Geoffroy; King, Tamara; Wang, Jing; Damaj, M Imad; Korczeniewska, Olga A; Camacho, Carlos J; Khanna, Rajesh

Late-Stage Modification of Oligopeptides by Nickel-Catalyzed Stereoselective Radical Addition to Dehydroalanine

镍催化脱氢丙氨酸立体选择性自由基加成反应对寡肽进行后期修饰

Qi, Xiaoxu; Jambu, Subramanian; Ji, Yining; Belyk, Kevin M; Panigrahi, Nihar R; Arora, Paramjit S; Strotman, Neil A; Diao, Tianning

Peptide Tethering: Pocket-Directed Fragment Screening for Peptidomimetic Inhibitor Discovery

肽链连接:用于发现肽模拟抑制剂的口袋导向片段筛选

Modell, Ashley E; Marrone, Frank 3rd; Panigrahi, Nihar R; Zhang, Yingkai; Arora, Paramjit S