日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel Pyrrolo[3,2- d]pyrimidine Compounds Target Mitochondrial and Cytosolic One-carbon Metabolism with Broad-spectrum Antitumor Efficacy

新型吡咯并[3,2-d]嘧啶化合物靶向线粒体和细胞浆一碳代谢,具有广谱抗肿瘤功效

Aamod S Dekhne, Khushbu Shah, Gregory S Ducker, Jade M Katinas, Jennifer Wong-Roushar, Md Junayed Nayeen, Arpit Doshi, Changwen Ning, Xun Bao, Josephine Frühauf, Jenney Liu, Adrianne Wallace-Povirk, Carrie O'Connor, Sijana H Dzinic, Kathryn White, Juiwanna Kushner, Seongho Kim, Maik Hüttemann, Lisa

AG311, a small molecule inhibitor of complex I and hypoxia-induced HIF-1α stabilization

AG311,一种复合物 I 的小分子抑制剂和缺氧诱导的 HIF-1α 稳定剂

Anja Bastian, Satoshi Matsuzaki, Kenneth M Humphries, Gavin A Pharaoh, Arpit Doshi, Nilesh Zaware, Aleem Gangjee, Michael A Ihnat