日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Venetoclax Penetrates the Blood Brain Barrier: A Pharmacokinetic Analysis in Pediatric Leukemia Patients

维奈托克可穿透血脑屏障:一项针对儿童白血病患者的药代动力学分析

Badawi, Mohamed; Menon, Rajeev; Place, Andrew E; Palenski, Tammy; Sunkersett, Gauri; Arrendale, Richard; Deng, Rong; Federico, Sara M; Cooper, Todd M; Salem, Ahmed Hamed

An orally available, small-molecule polymerase inhibitor shows efficacy against a lethal morbillivirus infection in a large animal model

一种口服的小分子聚合酶抑制剂在大动物模型中显示出对致命性麻疹病毒感染的疗效。

Krumm, Stefanie A; Yan, Dan; Hovingh, Elise S; Evers, Taylor J; Enkirch, Theresa; Reddy, G Prabhakar; Sun, Aiming; Saindane, Manohar T; Arrendale, Richard F; Painter, George; Liotta, Dennis C; Natchus, Michael G; von Messling, Veronika; Plemper, Richard K

Effect of protein binding on unbound atazanavir and darunavir cerebrospinal fluid concentrations

蛋白质结合对脑脊液中游离阿扎那韦和达芦那韦浓度的影响

Delille, Cecile A; Pruett, Sarah T; Marconi, Vincent C; Lennox, Jeffrey L; Armstrong, Wendy S; Arrendale, Richard F; Sheth, Anandi N; Easley, Kirk A; Acosta, Edward P; Vunnava, Aswani; Ofotokun, Ighovwerha

Discovery of tetrahydroisoquinoline-based CXCR4 antagonists

发现基于四氢异喹啉的CXCR4拮抗剂

Truax, Valarie M; Zhao, Huanyu; Katzman, Brooke M; Prosser, Anthony R; Alcaraz, Ana A; Saindane, Manohar T; Howard, Randy B; Culver, Deborah; Arrendale, Richard F; Gruddanti, Prahbakar R; Evers, Taylor J; Natchus, Michael G; Snyder, James P; Liotta, Dennis C; Wilson, Lawrence J

Development of a unique small molecule modulator of CXCR4

开发一种独特的CXCR4小分子调节剂

Liang, Zhongxing; Zhan, Weiqiang; Zhu, Aizhi; Yoon, Younghyoun; Lin, Songbai; Sasaki, Maiko; Klapproth, Jan-Michael A; Yang, Hua; Grossniklaus, Hans E; Xu, Jianguo; Rojas, Mauricio; Voll, Ronald J; Goodman, Mark M; Arrendale, Richard F; Liu, Jin; Yun, C Chris; Snyder, James P; Liotta, Dennis C; Shim, Hyunsuk

Synthesis of a phosphoserine mimetic prodrug with potent 14-3-3 protein inhibitory activity

合成一种具有强效14-3-3蛋白抑制活性的磷酸丝氨酸模拟前药

Arrendale, Allison; Kim, Keunho; Choi, Jun Young; Li, Wei; Geahlen, Robert L; Borch, Richard F

Synthetic curcumin analog EF31 inhibits the growth of head and neck squamous cell carcinoma xenografts

合成姜黄素类似物 EF31 抑制头颈部鳞状细胞癌异种移植瘤的生长

Shijun Zhu, Terry W Moore, Xiaoqian Lin, Nao Morii, Alessandra Mancini, Randy B Howard, Deborah Culver, Richard F Arrendale, Prabhakar Reddy, Taylor J Evers, Hongzheng Zhang, Gabriel Sica, Zhuo G Chen, Aiming Sun, Haian Fu, Fadlo R Khuri, Dong M Shin, James P Snyder, Mamoru Shoji

Assessment of glycated hemoglobin using A1CNow+ point-of-care device as compared to central laboratory testing

使用 A1CNow+ 即时检测设备评估糖化血红蛋白与中心实验室检测的比较

Arrendale, Justin R; Cherian, Sonia E; Zineh, Issam; Chirico, Mark J; Taylor, James R