日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The N-Myc MB0-MBI region interacts specifically and dynamically with the N-lobe of Aurora kinase A

N-Myc MB0-MBI 区与 Aurora 激酶 A 的 N 端结构域发生特异性且动态的相互作用。

Hultman, Johanna; Morad, Vivian; Tanner, Eliane; Kenney, Tristan M G; Pietras, Zuzanna; Khare, Lalit Pramod; Derbyshire, Dean; Resetca, Diana; Arrowsmith, Cheryl H; Aili, Daniel; Ekström, Simon; Penn, Linda Z; Wallner, Björn; Ahlner, Alexandra; Sunnerhagen, Maria

A synergistic interaction between PRMT5 and LSD1 inhibitors in AML.

PRMT5 和 LSD1 抑制剂在急性髓系白血病中存在协同作用。

Param Nesteene Joy, Arceci Elisa, Fiorentino Francesco, Pignata Luca, Torre Denis, Gutiérrez-Trejo Nayeli, Fong Jia Yi, Goy Pierre-Alexis, Han Brenda Y, Lambona Chiara, Di Bello Elisabetta, Castiello Carola, Barone Marco, Schwarz Megan, Arrowsmith Cheryl, Ito Koichi, Scherle Peggy, Wee Dave Keng Boon, Ndoye Steven, Tabaglio Tommaso, Jeyasekharan Anand D, Lakshmanan Manikandan, Cirilli Roberto, Habisch Hansjörg, Madl Tobias, Mattevi Andrea, Valente Sergio, Mai Antonello, Guccione Ernesto

CACHE Challenge #3: Targeting the Nsp3 Macrodomain of SARS-CoV-2

CACHE挑战赛#3:靶向SARS-CoV-2的Nsp3宏结构域

Herasymenko, Oleksandra; Silva, Madhushika; Correy, Galen J; Abu-Saleh, Abd Al-Aziz A; Ackloo, Suzanne; Arrowsmith, Cheryl; Ashworth, Alan; Ban, Fuqiang; Beck, Hartmut; Bishop, Kevin P; Bohórquez, Hugo J; Bolotokova, Albina; Breznik, Marko; Chau, Irene; Chen, Yu; Cherkasov, Artem; Dehaen, Wim; Della Corte, Dennis; Denzinger, Katrin; Doering, Niklas P; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Gentile, Francesco; Gibson, Elisa; Gokdemir, Ozan; Gunnarsson, Anders; Günther, Judith; Irwin, John J; Jensen, Jan Halborg; Harding, Rachel J; Hillisch, Alexander; Hoffer, Laurent; Hogner, Anders; Hutchinson, Ashley; Kandwal, Shubhangi; Karlova, Andrea; Koirala, Kushal; Kotelnikov, Sergei; Kozakov, Dima; Lee, Juyong; Lee, Soowon; Lessel, Uta; Liu, Sijie; Liu, Xuefeng; Loppnau, Peter; Meiler, Jens; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Oprea, Tudor I; Paige, Brooks; Pandit, Amit; Park, Keunwan; Poda, Gennady; Protopopov, Mykola V; Pütter, Vera; Ravichandran, Rahul; Rognan, Didier; Rosta, Edina; Sabnis, Yogesh; Scott, Thomas; Seitova, Almagul; Sharma, Purshotam; Sindt, François; Song, Minghu; Steinmann, Casper; Stevens, Rick; Talagayev, Valerij; Tararina, Valentyna V; Tarkhanova, Olga; Tingey, Damon; Trant, John F; Treleaven, Dakota; Tropsha, Alexander; Walters, Patrick; Wells, Jude; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zheng, Shuangjia; Fraser, James S; Schapira, Matthieu

Glioblastoma stem cells show transcriptionally correlated spatial organization

胶质母细胞瘤干细胞表现出转录相关的空间组织结构

Ayyadhury, Shamini; Sachamitr, Patty; Kushida, Michelle M; Park, Nicole I; Coutinho, Fiona J; Whitley, Owen; Prinos, Panagiotis; Arrowsmith, Cheryl H; Dirks, Peter B; Pugh, Trevor J; Bader, Gary D

A needed nomenclature for nucleosomes

核小体命名法的必要性

Keogh, Michael-Christopher; Almouzni, Genevieve; Andrews, Andrew J; Armache, Karim-Jean; Arrowsmith, Cheryl H; Baek, Sung Hee; Bedford, Mark T; Bernstein, Emily; Côté, Jacques; David, Yael; Denu, John M; Fierz, Beat; Garcia, Benjamin A; Glass, Karen C; Gozani, Or; Helin, Kristian; Henikoff, Steven; Jensen, Ole N; Josefowicz, Steven Z; Kelleher, Neil L; Kutateladze, Tatiana G; Lindner, Herbert H; Lu, Chao; Luger, Karolin; Mallick, Parag; Musselman, Catherine A; Muir, Tom W; Paša-Tolić, Ljiljana; Schneider, Robert; Shi, Xiaobing; Shi, Yang; Sidoli, Simone; Smith, Lloyd M; Tyler, Jessica K; Wolberger, Cynthia; Workman, Jerry L; Strahl, Brian D; Young, Nicolas L

Enantioselective protein affinity selection mass spectrometry (E-ASMS)

对映选择性蛋白质亲和力选择质谱法(E-ASMS)

Wang, Xiaoyun; Sun, Jianxian; Ahmad, Shabbir; Yang, Diwen; Li, Fengling; Chan, U Hang; Zeng, Hong; Simoben, Conrad V; Green, Stuart R; Silva, Madhushika; Houliston, Scott; Dong, Aiping; Bolotokova, Albina; Gibson, Elisa; Kutera, Maria; Ghiabi, Pegah; Kondratov, Ivan; Matviyuk, Tetiana; Chuprina, Alexander; Mavridi, Danai; Lenz, Christopher; Joerger, Andreas C; Brown, Benjamin D; Heath, Richard B; Yue, Wyatt W; Robbie, Lucy K; Beyett, Tyler S; Müller, Susanne; Knapp, Stefan; Owen, Dafydd R; Harding, Rachel; Schapira, Matthieu; Brown, Peter J; Santhakumar, Vijayaratnam; Ackloo, Suzanne; Arrowsmith, Cheryl H; Edwards, Aled M; Peng, Hui; Halabelian, Levon

Characterization of PROTAC specificity and endogenous protein interactomes using ProtacID.

利用ProtacID对PROTAC特异性和内源性蛋白质相互作用组进行表征

Shrestha Suman, Maitland Matthew E R, Jing Laili, Duan Shili, Nie David Y, St-Germain Jonathan, Kanaris Michael, Barsyte-Lovejoy Dalia, Arrowsmith Cheryl H, Raught Brian

Structural basis of TMPRSS11D specificity and autocleavage activation.

TMPRSS11D 特异性和自切割激活的结构基础

Fraser Bryan J, Wilson Ryan P, Ferková Sára, Ilyassov Olzhas, Lac Jackie, Dong Aiping, Li Yen-Yen, Seitova Alma, Li Yanjun, Hejazi Zahra, Kenney Tristan M G, Penn Linda Z, Edwards Aled, Leduc Richard, Boudreault Pierre-Luc, Morin Gregg B, Bénard François, Arrowsmith Cheryl H

PRMT5 promotes full-length HTT expression by repressing multiple proximal intronic polyadenylation sites.

PRMT5 通过抑制多个近端内含子多聚腺苷酸化位点来促进全长 HTT 表达

Yadav Manisha, AlQazzaz Mona A, Ciamponi Felipe E, Ho Jolene C, Maron Maxim I, Sababi Aiden M, MacLeod Graham, Ahmadi Moloud, Bullivant Garrett, Tano Vincent, Langley Sarah R, Sánchez-Osuna María, Sachamitr Patty, Kushida Michelle, Bardile Costanza Ferrari, Pouladi Mahmoud A, Kurtz Rebecca, Richards Laura, Pugh Trevor, Tyers Mike, Angers Stephane, Dirks Peter B, Bader Gary D, Truant Ray, Massirer Katlin B, Barsyte-Lovejoy Dalia, Shechter David, Harding Rachel J, Arrowsmith Cheryl H, Prinos Panagiotis

Serine phosphorylation facilitates protein degradation by the human mitochondrial ClpXP protease

丝氨酸磷酸化促进人线粒体ClpXP蛋白酶对蛋白质的降解

Feng, Yue; Goncalves, Monica M; Jitkova, Yulia; Keszei, Alexander F A; Yan, Yongran; Sarathy, Chaitra; St-Germain, Jonathan; Kenney, Tristan M G; Tcheng, Matthew; Trudel, Vincent; Mancini, Ross S; Upadhyay, Rahul; Hurren, Rose; Gronda, Marcela; Schultz, Matthew; Soriano, Kaylen; Lees, Kaitlin; Pomroy, Neil C; Currie, S Quinn W; Privé, Gilbert G; Reed, Mark A; Yudin, Andrei K; Penn, Linda Z; Arrowsmith, Cheryl H; Raught, Brian; Mazhab-Jafari, Mohammad T; Vahidi, Siavash; Schimmer, Aaron D