High-resolution deep mutational scanning of the melanocortin-4 receptor enables target characterization for drug discovery
对黑皮质素-4受体进行高分辨率深度突变扫描,能够实现药物发现的靶点表征。
期刊:Elife
影响因子:6.4
doi:10.7554/eLife.104725
Howard, Conor J; Abell, Nathan S; Osuna, Beatriz A; Jones, Eric M; Chan, Leon Y; Chan, Henry; Artis, Dean R; Asfaha, Jonathan B; Bloom, Joshua S; Cooper, Aaron R; Liao, Andrew; Mahdavi, Eden; Mohammed, Nabil; Su, Alan L; Uribe, Giselle A; Kosuri, Sriram; Dickel, Diane E; Lubock, Nathan B