日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Small-molecule inhibition of METTL3 as a strategy against myeloid leukaemia

小分子抑制剂METTL3作为对抗髓系白血病的策略

Eliza Yankova # ,Wesley Blackaby # ,Mark Albertella ,Justyna Rak ,Etienne De Braekeleer ,Georgia Tsagkogeorga ,Ewa S Pilka ,Demetrios Aspris ,Dan Leggate ,Alan G Hendrick ,Natalie A Webster ,Byron Andrews ,Richard Fosbeary ,Patrick Guest ,Nerea Irigoyen ,Maria Eleftheriou ,Malgorzata Gozdecka ,Joao M L Dias ,Andrew J Bannister ,Binje Vick ,Irmela Jeremias ,George S Vassiliou ,Oliver Rausch ,Konstantinos Tzelepis ,Tony Kouzarides

METTL1-mediated m7G modification of Arg-TCT tRNA drives oncogenic transformation

METTL1 介导的 Arg-TCT tRNA 的 m7G 修饰驱动致癌转化

Esteban A Orellana, Qi Liu, Eliza Yankova, Mehdi Pirouz, Etienne De Braekeleer, Wencai Zhang, Jihoon Lim, Demetrios Aspris, Erdem Sendinc, Dimitrios A Garyfallos, Muxin Gu, Raja Ali, Alejandro Gutierrez, Sigitas Mikutis, Gonçalo J L Bernardes, Eric S Fischer, Allan Bradley, George S Vassiliou, Frank

The N6-methyladenosine RNA modification in acute myeloid leukemia

急性髓系白血病中的N6-甲基腺苷RNA修饰

Yankova, Eliza; Aspris, Demetrios; Tzelepis, Konstantinos

meCLICK-Seq, a Substrate-Hijacking and RNA Degradation Strategy for the Study of RNA Methylation

meCLICK-Seq:一种用于研究RNA甲基化的底物劫持和RNA降解策略

Sigitas Mikutis ,Muxin Gu ,Erdem Sendinc ,Madoka E Hazemi ,Hannah Kiely-Collins ,Demetrios Aspris ,George S Vassiliou ,Yang Shi ,Konstantinos Tzelepis ,Gonçalo J L Bernardes

SRPK1 maintains acute myeloid leukemia through effects on isoform usage of epigenetic regulators including BRD4

SRPK1通过影响包括BRD4在内的表观遗传调控因子的亚型使用来维持急性髓系白血病。

Konstantinos Tzelepis ,Etienne De Braekeleer ,Demetrios Aspris ,Isaia Barbieri ,M S Vijayabaskar ,Wen-Hsin Liu ,Malgorzata Gozdecka ,Emmanouil Metzakopian ,Hamish D Toop ,Monika Dudek ,Samuel C Robson ,Francisco Hermida-Prado ,Yu Hsuen Yang ,Roya Babaei-Jadidi ,Dimitrios A Garyfallos ,Hannes Ponstingl ,Joao M L Dias ,Paolo Gallipoli ,Michael Seiler ,Silvia Buonamici ,Binje Vick ,Andrew J Bannister ,Roland Rad ,Rab K Prinjha ,John C Marioni ,Brian Huntly ,Jennifer Batson ,Jonathan C Morris ,Cristina Pina ,Allan Bradley ,Irmela Jeremias ,David O Bates ,Kosuke Yusa ,Tony Kouzarides ,George S Vassiliou

Promoter-bound METTL3 maintains myeloid leukaemia by m6A-dependent translation control

启动子结合的METTL3通过m6A依赖性翻译调控维持髓系白血病。

Isaia Barbieri ,Konstantinos Tzelepis ,Luca Pandolfini ,Junwei Shi ,Gonzalo Millán-Zambrano ,Samuel C Robson ,Demetrios Aspris ,Valentina Migliori ,Andrew J Bannister ,Namshik Han ,Etienne De Braekeleer ,Hannes Ponstingl ,Alan Hendrick ,Christopher R Vakoc ,George S Vassiliou ,Tony Kouzarides