日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

BRF110, an Orally Active Nurr1-RXRα-Selective Rexinoid, Enhances BDNF Expression without Elevating Triglycerides

BRF110 是一种口服活性 Nurr1-RXRα 选择性雷西诺类药物,可在不升高甘油三酯的情况下增强 BDNF 表达。

Xenophon Asvos,Mohamed A El Mubarak,Theodoros Karampelas,Theodoros Rampias,Constantin Tamvakopoulos,Gregory B Sivolapenko,Athanasios Papakyriakou,Stavros Topouzis,Demetrios K Vassilatis,Demosthenes Fokas

Polymorphic positions 349 and 725 of the autoimmunity-protective allotype 10 of ER aminopeptidase 1 are key in determining its unique enzymatic properties

ER 氨基肽酶 1 的自身免疫保护同种型 10 的多态性位置 349 和 725 是决定其独特酶特性的关键

Galateia Georgaki, Anastasia Mpakali, Myrto Trakada, Athanasios Papakyriakou, Efstratios Stratikos

Structure-Based Discovery of Receptor Activator of Nuclear Factor-κB Ligand (RANKL)-Induced Osteoclastogenesis Inhibitors

基于结构发现核因子 κB 受体激活剂配体 (RANKL) 诱导的破骨细胞生成抑制剂

Vagelis Rinotas, Fotini Liepouri, Maria-Dimitra Ouzouni, Niki Chalkidi, Christos Papaneophytou, Mariza Lampropoulou, Veroniki P Vidali, George Kontopidis, Elias Couladouros, Elias Eliopoulos, Athanasios Papakyriakou, Eleni Douni

The Inhibitory Properties of a Novel, Selective LMTK3 Kinase Inhibitor

新型选择性 LMTK3 激酶抑制剂的抑制特性

Alessandro Agnarelli, Andrea Lauer Betrán, Athanasios Papakyriakou, Viviana Vella, Mark Samuels, Panagiotis Papanastasopoulos, Christina Giamas, Erika J Mancini, Justin Stebbing, John Spencer, Chiara Cilibrasi, Angeliki Ditsiou, Georgios Giamas

Design, synthesis and biological evaluation of new 3,4-dihydroquinoxalin-2(1 H)-one derivatives as soluble guanylyl cyclase (sGC) activators

新型 3,4-二氢喹喔啉-2(1H)-酮衍生物作为可溶性鸟苷酸环化酶 (sGC) 激活剂的设计、合成及生物学评价

Dionysios-Panagiotis Kintos, Konstantinos Salagiannis, Vasiliki Vazoura, Theresa Wittrien, Athanasios Papakyriakou, Sotiris S Nikolaropoulos, Soenke Behrends, Stavros Topouzis, Manolis A Fousteris

5-ALA Is a Potent Lactate Dehydrogenase Inhibitor but Not a Substrate: Implications for Cell Glycolysis and New Avenues in 5-ALA-Mediated Anticancer Action

5-ALA 是一种有效的乳酸脱氢酶抑制剂,但不是底物:对细胞糖酵解的影响以及 5-ALA 介导的抗癌作用的新途径

Mantas Grigalavicius, Somayeh Ezzatpanah, Athanasios Papakyriakou, Tine Therese Henriksen Raabe, Konstantina Yannakopoulou, Theodossis A Theodossiou

The structure-function relationship of oncogenic LMTK3

致癌基因 LMTK3 的结构与功能关系

Angeliki Ditsiou, Chiara Cilibrasi, Nikiana Simigdala, Athanasios Papakyriakou, Leanne Milton-Harris, Viviana Vella, Joanne E Nettleship, Jae Ho Lo, Shivani Soni, Goar Smbatyan, Panagiota Ntavelou, Teresa Gagliano, Maria Chiara Iachini, Sahir Khurshid, Thomas Simon, Lihong Zhou, Storm Hassell-Hart, 

Discovery of Small-Molecule Inhibitors of Receptor Activator of Nuclear Factor-κB Ligand with a Superior Therapeutic Index

发现具有优异治疗指数的核因子-κB受体激活剂配体小分子抑制剂

Vagelis Rinotas, Athanasios Papakyriakou, Foteini Violitzi, Christos Papaneophytou, Maria-Dimitra Ouzouni, Polyxeni Alexiou, Alexandros Strongilos, Elias Couladouros, George Kontopidis, Elias Eliopoulos, Eleni Douni

A systematic re-examination of processing of MHCI-bound antigenic peptide precursors by endoplasmic reticulum aminopeptidase 1

系统地重新检查内质网氨基肽酶 1 对 MHCI 结合抗原肽前体的加工

George Mavridis, Richa Arya, Alexander Domnick, Jerome Zoidakis, Manousos Makridakis, Antonia Vlahou, Anastasia Mpakali, Angelos Lelis, Dimitris Georgiadis, Robert Tampé, Athanasios Papakyriakou, Lawrence J Stern, Efstratios Stratikos

Editing the immunopeptidome of melanoma cells using a potent inhibitor of endoplasmic reticulum aminopeptidase 1 (ERAP1)

使用内质网氨基肽酶 1 (ERAP1) 的强效抑制剂编辑黑色素瘤细胞的免疫肽组

Despoina Koumantou, Eilon Barnea, Adrian Martin-Esteban, Zachary Maben, Athanasios Papakyriakou, Anastasia Mpakali, Paraskevi Kokkala, Harris Pratsinis, Dimitris Georgiadis, Lawrence J Stern, Arie Admon, Efstratios Stratikos