日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The BTK Inhibitor Ibrutinib (PCI-32765) Overcomes Paclitaxel Resistance in ABCB1- and ABCC10-Overexpressing Cells and Tumors

BTK 抑制剂 Ibrutinib (PCI-32765) 可克服 ABCB1 和 ABCC10 过表达细胞和肿瘤中的紫杉醇耐药性

Hui Zhang, Atish Patel, Yi-Jun Wang, Yun-Kai Zhang, Rishil J Kathawala, Long-Hui Qiu, Bhargav A Patel, Li-Hua Huang, Suneet Shukla, Dong-Hua Yang, Suresh V Ambudkar, Li-Wu Fu, Zhe-Sheng Chen

Revealing the fate of cell surface human P-glycoprotein (ABCB1): The lysosomal degradation pathway

揭示细胞表面人类 P-糖蛋白 (ABCB1) 的命运:溶酶体降解途径

Kazuhiro Katayama, Khyati Kapoor, Shinobu Ohnuma, Atish Patel, William Swaim, Indu S Ambudkar, Suresh V Ambudkar

A-803467, a tetrodotoxin-resistant sodium channel blocker, modulates ABCG2-mediated MDR in vitro and in vivo

A-803467 是一种抗河豚毒素钠通道阻滞剂,可在体内和体外调节 ABCG2 介导的 MDR

Nagaraju Anreddy, Atish Patel, Yun-Kai Zhang, Yi-Jun Wang, Suneet Shukla, Rishil J Kathawala, Priyank Kumar, Pranav Gupta, Suresh V Ambudkar, John N D Wurpel, Zhe-Sheng Chen, Huiqin Guo

IKK inhibition increases bortezomib effectiveness in ovarian cancer

IKK 抑制可增强硼替佐米治疗卵巢癌的疗效

Bipradeb Singha, Himavanth Reddy Gatla, Sai Phyo, Atish Patel, Zhe-Sheng Chen, Ivana Vancurova

The small molecule tyrosine kinase inhibitor NVP-BHG712 antagonizes ABCC10-mediated paclitaxel resistance: a preclinical and pharmacokinetic study

小分子酪氨酸激酶抑制剂 NVP-BHG712 拮抗 ABCC10 介导的紫杉醇耐药性:临床前和药代动力学研究

Rishil J Kathawala, Liuya Wei, Nagaraju Anreddy, Kang Chen, Atish Patel, Saeed Alqahtani, Yun-Kai Zhang, Yi-Jun Wang, Kamlesh Sodani, Amal Kaddoumi, Charles R Ashby Jr, Zhe-Sheng Chen

PD173074, a selective FGFR inhibitor, reverses MRP7 (ABCC10)-mediated MDR

PD173074 是一种选择性 FGFR 抑制剂,可逆转 MRP7 (ABCC10) 介导的 MDR

Nagaraju Anreddy, Atish Patel, Kamlesh Sodani, Rishil J Kathawala, Eugenie P Chen, John N D Wurpel, Zhe-Sheng Chen

In vitro, in vivo and ex vivo characterization of ibrutinib: a potent inhibitor of the efflux function of the transporter MRP1

依鲁替尼的体外、体内和离体表征:转运蛋白 MRP1 外排功能的强效抑制剂

Hui Zhang, Atish Patel, Shao-Lin Ma, Xiao Jie Li, Yun-Kai Zhang, Pei-Qi Yang, Rishil J Kathawala, Yi-Jun Wang, Nagaraju Anreddy, Li-Wu Fu, Zhe-Sheng Chen

Telatinib reverses chemotherapeutic multidrug resistance mediated by ABCG2 efflux transporter in vitro and in vivo

替拉替尼在体内和体外逆转由 ABCG2 外排转运体介导的化疗多药耐药性

Kamlesh Sodani, Atish Patel, Nagaraju Anreddy, Satyakam Singh, Dong-Hua Yang, Rishil J Kathawala, Priyank Kumar, Tanaji T Talele, Zhe-Sheng Chen

Masitinib antagonizes ATP-binding cassette subfamily C member 10-mediated paclitaxel resistance: a preclinical study

马赛替尼拮抗 ATP 结合盒亚家族 C 成员 10 介导的紫杉醇耐药性:一项临床前研究

Rishil J Kathawala, Kamlesh Sodani, Kang Chen, Atish Patel, Alaa H Abuznait, Nagaraju Anreddy, Yue-Li Sun, Amal Kaddoumi, Charles R Ashby Jr, Zhe-Sheng Chen

WHI-P154 enhances the chemotherapeutic effect of anticancer agents in ABCG2-overexpressing cells

WHI-P154 增强抗癌药物在 ABCG2 过表达细胞中的化疗效果

Hui Zhang, Yun-Kai Zhang, Yi-Jun Wang, Rishil J Kathawala, Atish Patel, Hua Zhu, Kamlesh Sodani, Tanaji T Talele, Suresh V Ambudkar, Zhe-Sheng Chen, Li-Wu Fu