日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, synthesis, and anticancer activity of novel isocryptolepine 'aza' type acyl thiourea derivatives via combined experimental and computational approach

通过实验和计算相结合的方法设计、合成新型异隐花碱“氮杂”型酰基硫脲衍生物及其抗癌活性

Fayyaz, Ammara; Ejaz, Syeda Abida; Ahmed, Atteeque; Channar, Pervaiz Ali; Afzal, Saira; Ujan, Rabail; Saeed, Aamer; Bibi, Rifhat; Alsfouk, Bshra A; Abbas, Qamar; Sahito, Reshma; Bolte, Michael; Hökelek, Tuncer

Synthesis and evaluation of thiazolyl coumarin drug conjugates as carbonic anhydrase isozyme inhibitors by using integrated invitro and insilico approaches

利用体外和计算机模拟相结合的方法合成和评价噻唑基香豆素药物偶联物作为碳酸酐酶同工酶抑制剂的活性

Ahmed, Atteeque; Kanwal, Romaisa; Channar, Pervaiz Ali; Alshahrani, Mohammad Y; Saeed, Aamer; Ejaz, Syeda Abida; Attaullah, Hafiz Muhammad; Bibi, Rifhat; Li, Chen

Discovery of isatin-thiazole conjugates as potent urease inhibitors; synthesis, biochemical screening and computational studies

发现靛红-噻唑缀合物作为强效脲酶抑制剂;合成、生化筛选和计算研究

Haider, Mian Bilal; Zaib, Sumera; Saeed, Aamer; Ahmed, Atteeque; Javed, Hira; Areeba; Shabir, Ghulam; Irfan, Madiha; Othman, Gehan Ahmed

Novel pyrazoline linked acyl thiourea pharmacophores as antimicrobial, urease, amylase and α-glucosidase inhibitors: design, synthesis, SAR and molecular docking studies

新型吡唑啉连接的酰基硫脲药效团作为抗菌、脲酶、淀粉酶和α-葡萄糖苷酶抑制剂:设计、合成、构效关系和分子对接研究

Saeed, Aamer; Ahmed, Atteeque; Haider, Main Bilal; Ismail, Hammad; Hayat, Khizar; Shabir, Ghulam; El-Seedi, Hesham R

Acyl pyrazole sulfonamides as new antidiabetic agents: synthesis, glucosidase inhibition studies, and molecular docking analysis

酰基吡唑磺酰胺类化合物作为新型抗糖尿病药物:合成、葡萄糖苷酶抑制研究及分子对接分析

Ahmed, Atteeque; Zaib, Sumera; Bhat, Mashooq Ahmad; Saeed, Aamer; Altaf, Muhammad Zain; Zahra, Fatima Tuz; Shabir, Ghulam; Rana, Nehal; Khan, Imtiaz

Synthesis of amantadine clubbed N-aryl amino thiazoles as potent urease, α-amylase & α-glucosidase inhibitors, kinetic and molecular docking studies

合成金刚烷胺偶联的N-芳基氨基噻唑类化合物作为强效脲酶、α-淀粉酶和α-葡萄糖苷酶抑制剂,并进行动力学和分子对接研究

Zahra, Fatima Tuz; Saeed, Aamer; Ahmed, Atteeque; Ismail, Hammad; Ijaz, Muhammad Umar; Albericio, Fernando

Novel adamantyl clubbed iminothiazolidinones as promising elastase inhibitors: design, synthesis, molecular docking, ADMET and DFT studies

新型金刚烷基亚氨基噻唑烷酮作为有前途的弹性蛋白酶抑制剂:设计、合成、分子对接、ADMET 和 DFT 研究

Atteeque Ahmed, Aamer Saeed, Syeda Abida Ejaz, Mubashir Aziz, Muhammad Zaffar Hashmi, Pervaiz Ali Channar, Qamar Abbas, Hussain Raza, Zahid Shafiq, Hesham R El-Seedi