日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

ABBV-011, A Novel, Calicheamicin-Based Antibody-Drug Conjugate, Targets SEZ6 to Eradicate Small Cell Lung Cancer Tumors

ABBV-011 是一种新型基于卡里车霉素的抗体-药物偶联物,靶向 SEZ6 以根除小细胞肺癌肿瘤

Wolf R Wiedemeyer, Julia Gavrilyuk, Alexander Schammel, Xi Zhao, Hetal Sarvaiya, Marybeth Pysz, Christine Gu, Monica You, Kumiko Isse, Theodore Sullivan, Dorothy French, Christina Lee, Angeline T Dang, Zhaomei Zhang, Monette Aujay, Alexander J Bankovich, Philip Vitorino

Uncialamycin-based antibody-drug conjugates: Unique enediyne ADCs exhibiting bystander killing effect

基于安西拉霉素的抗体药物偶联物:具有旁观者杀伤效应的独特烯二炔类抗体药物偶联物

Nicolaou, K C; Rigol, Stephan; Pitsinos, Emmanuel N; Das, Dipendu; Lu, Yong; Rout, Subhrajit; Schammel, Alexander W; Holte, Dane; Lin, Baiwei; Gu, Christine; Sarvaiya, Hetal; Trinidad, Jose; Barbour, Nicole; Valdiosera, Amanda M; Sandoval, Joseph; Lee, Christina; Aujay, Monette; Fernando, Hanan; Dhar, Anukriti; Karsunky, Holger; Taylor, Nicole; Pysz, Marybeth; Gavrilyuk, Julia

A DLL3-targeted antibody-drug conjugate eradicates high-grade pulmonary neuroendocrine tumor-initiating cells in vivo

DLL3 靶向抗体-药物偶联物可在体内清除高级别肺神经内分泌肿瘤起始细胞

Laura R Saunders, Alexander J Bankovich, Wade C Anderson, Monette A Aujay, Sheila Bheddah, KristenAnn Black, Radhika Desai, Paul A Escarpe, Johannes Hampl, Amy Laysang, David Liu, Javier Lopez-Molina, Milly Milton, Albert Park, Marybeth A Pysz, Hui Shao, Brian Slingerland, Michael Torgov, Samuel A W

Synergistic effects of proteasome inhibitor carfilzomib in combination with tyrosine kinase inhibitors in imatinib-sensitive and -resistant chronic myeloid leukemia models

蛋白酶体抑制剂卡非佐米与酪氨酸激酶抑制剂联合用于伊马替尼敏感和耐药慢性粒细胞白血病模型的协同作用

L J Crawford, E T Chan, M Aujay, T L Holyoake, J V Melo, H G Jorgensen, S Suresh, B Walker, A E Irvine

PR-924, a selective inhibitor of the immunoproteasome subunit LMP-7, blocks multiple myeloma cell growth both in vitro and in vivo

PR-924 是一种选择性免疫蛋白酶体亚基 LMP-7 抑制剂,可在体外和体内抑制多发性骨髓瘤细胞的生长。

Singh, Ajita V; Bandi, Madhavi; Aujay, Monette A; Kirk, Christopher J; Hark, David E; Raje, Noopur; Chauhan, Dharminder; Anderson, Kenneth C