日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of potent inhibitors of Leishmania donovani and Leishmania infantum chagasi, the causative agents of Old and New World visceral leishmaniasis

鉴定出能有效抑制杜氏利什曼原虫和婴儿利什曼原虫(旧大陆和新大陆内脏利什曼病病原体)的药物

Zulfiqar, Bilal; Colombo, Fabio Antonio; Nunes, Juliana Barbosa; Espuri, Patricia Ferreira; Ferreira, Aurea Favero; Manthri, Sujatha; De Rycker, Manu; Marques, Marcos Jose; Avery, Vicky M

Heterocyclic core modifications in trypanosomacidal 2-[(phenylheteroaryl)ethyl]ureas

锥虫杀灭剂 2-[(苯基杂芳基)乙基]脲的杂环核心修饰

Toynton, Arthur; Ferrins, Lori; Newson, Harriet L; Sykes, Melissa L; Varghese, Swapna; Nguyen, Nghi; Russell, Stephanie; Rahmani, Raphaël; Cheang, Jeremy; Flematti, Gavin R; Skelton, Brian W; Zulfiqar, Bilal; Avery, Vicky M; Baell, Jonathan B; Piggott, Matthew J

S-MGBs bearing amidine tail groups are potent, selective antiplasmodial agents.

带有脒基尾部的 S-MGB 是强效、选择性的抗疟原虫药物

Perieteanu Marina, Garzon Tayner Rodriguez, McGee Leah M C, Khalaf Abedawn I, Suckling Colin J, Beveridge Rebecca, Avery Vicky M, Scott Fraser J

DNDI-6174 is a preclinical candidate for visceral leishmaniasis that targets the cytochrome bc(1)

DNDI-6174 是一种用于治疗内脏利什曼病的临床前候选药物,其靶点为细胞色素 bc(1)

Braillard, Stéphanie; Keenan, Martine; Breese, Karen J; Heppell, Jacob; Abbott, Michael; Islam, Rafiqul; Shackleford, David M; Katneni, Kasiram; Crighton, Elly; Chen, Gong; Patil, Rahul; Lee, Given; White, Karen L; Carvalho, Sandra; Wall, Richard J; Chemi, Giulia; Zuccotto, Fabio; González, Silvia; Marco, Maria; Deakyne, Julianna; Standing, David; Brunori, Gino; Lyon, Jonathan J; Castañeda-Casado, Pablo; Camino, Isabel; Martinez Martinez, Maria S; Zulfiqar, Bilal; Avery, Vicky M; Feijens, Pim-Bart; Van Pelt, Natascha; Matheeussen, An; Hendrickx, Sarah; Maes, Louis; Caljon, Guy; Yardley, Vanessa; Wyllie, Susan; Charman, Susan A; Chatelain, Eric

Impact of Laboratory-Adapted Intracellular Trypanosoma cruzi Strains on the Activity Profiles of Compounds with Anti-T. cruzi Activity

实验室适应的细胞内锥虫株对具有抗克氏锥虫活性的化合物活性谱的影响

Sykes, Melissa L; Kennedy, Emily K; Avery, Vicky M

Temporal and Wash-Out Studies Identify Medicines for Malaria Venture Pathogen Box Compounds with Fast-Acting Activity against Both Trypanosoma cruzi and Trypanosoma brucei

时间序列和洗脱试验鉴定出疟疾风险病原体库化合物,这些化合物对克氏锥虫和布氏锥虫均具有快速活性。

Sykes, Melissa L; Kennedy, Emily K; Read, Kevin D; Kaiser, Marcel; Avery, Vicky M

Naturally Acquired Kelch13 Mutations in Plasmodium falciparum Strains Modulate In Vitro Ring-Stage Artemisinin-Based Drug Tolerance and Parasite Survival in Response to Hyperoxia

恶性疟原虫株中自然获得的 Kelch13 突变可调节体外环状体对青蒿素类药物的耐受性以及寄生虫在高氧条件下的存活率

Duffy, Sandra; Avery, Vicky M

The Novel bis-1,2,4-Triazine MIPS-0004373 Demonstrates Rapid and Potent Activity against All Blood Stages of the Malaria Parasite

新型双-1,2,4-三嗪化合物MIPS-0004373对疟原虫所有血液阶段均表现出快速而强效的活性

Ellis, Katherine M; Lucantoni, Leonardo; Chavchich, Marina; Abraham, Matthew; De Paoli, Amanda; Luth, Madeline R; Zeeman, Anne-Marie; Delves, Michael J; Terán, Fernando Sánchez-Román; Straschil, Ursula; Baum, Jake; Kocken, Clemens H M; Ralph, Stuart A; Winzeler, Elizabeth A; Avery, Vicky M; Edstein, Michael D; Baell, Jonathan B; Creek, Darren J

Antitubercular and Antiparasitic 2-Nitroimidazopyrazinones with Improved Potency and Solubility

具有增强的抗结核和抗寄生虫活性的2-硝基咪唑并吡嗪酮

Ang, Chee Wei; Tan, Lendl; Sykes, Melissa L; AbuGharbiyeh, Neda; Debnath, Anjan; Reid, Janet C; West, Nicholas P; Avery, Vicky M; Cooper, Matthew A; Blaskovich, Mark A T

Metabolic Roles of Androgen Receptor and Tip60 in Androgen-Dependent Prostate Cancer

雄激素受体和Tip60在雄激素依赖性前列腺癌中的代谢作用

Tan, Kah Ni; Avery, Vicky M; Carrasco-Pozo, Catalina