日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Heterodimeric JAK-STAT activation as a mechanism of persistence to JAK2 inhibitor therapy

异二聚体 JAK-STAT 激活是 JAK2 抑制剂治疗持续性的机制

Priya Koppikar, Neha Bhagwat, Outi Kilpivaara, Taghi Manshouri, Mazhar Adli, Todd Hricik, Fan Liu, Lindsay M Saunders, Ann Mullally, Omar Abdel-Wahab, Laura Leung, Abby Weinstein, Sachie Marubayashi, Aviva Goel, Mithat Gönen, Zeev Estrov, Benjamin L Ebert, Gabriela Chiosis, Stephen D Nimer, Bradley

Modulation of activation-loop phosphorylation by JAK inhibitors is binding mode dependent

JAK 抑制剂对活化环磷酸化的调节依赖于结合模式

Rita Andraos #, Zhiyan Qian #, Débora Bonenfant, Joëlle Rubert, Eric Vangrevelinghe, Clemens Scheufler, Fanny Marque, Catherine H Régnier, Alain De Pover, Hugues Ryckelynck, Neha Bhagwat, Priya Koppikar, Aviva Goel, Lorenza Wyder, Gisele Tavares, Fabienne Baffert, Carole Pissot-Soldermann, Paul W Ma