Linker substitution influences succinimide ring hydrolysis equilibrium impacting the stability of attachment to antibody-drug conjugates
连接基取代会影响琥珀酰亚胺环水解平衡,从而影响抗体-药物偶联物的连接稳定性。
期刊:RSC Medicinal Chemistry
影响因子:3.6
doi:10.1039/d3md00569k
Wang, Lu; Hobson, Adrian D; Salomon, Paulin L; Fitzgibbons, Julia; Xu, Jianwen; McCarthy, Sean; Wu, Kan; Jia, Ying; Hernandez, Axel Jr; Li, Xiang; Xu, Zhou; Wang, Zhongyuan; Yu, Yajie; Li, Junxian; Tao, Lin