日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Advances in BRET probes for intracellular target engagement studies

用于细胞内靶标结合研究的BRET探针的进展

Capener, Jacob L; Schwalm, Martin P; Vasta, James D; Michaud, Ani; Teske, Kelly A; Marsiglia, William M; Huber, Kilian V M; Dar, Arvin C; Knapp, Stefan; Axtman, Alison D; Robers, Matthew B

Development of a Chemical Probe to Enable Characterization of the Casein Kinase 1γ Subfamily

开发一种化学探针以实现酪蛋白激酶1γ亚家族的表征

Capener, Jacob L; Kramer, Thomas W; Bashore, Frances M; Flory, Emily; Li, Fengling; Strang, Blair L; Axtman, Alison D

Identification and optimization of first-in-class RNA helicase inhibitors of DDX1, LGP2, and MDA5

鉴定和优化首创的DDX1、LGP2和MDA5 RNA解旋酶抑制剂

Wang, Xiaowen; Wang, Feijun; Kong, Deyu; Uredi, Dilipkumar; Li, Fengling; Li, Feng; Rayadurgam, Jayachandra; Li, Hanxuan; Wolf, Esther; Chan, U Hang; Chau, Irene; Zeng, Hong; Perez, Julia Garcia; Wilson, Derek J; Bashore, Frances M; Wang, Xiaodong; Halabelian, Levon; Frankowski, Kevin J; Kireev, Dmitri; Axtman, Alison D

Targeting Na(v)1.7 and Na(v)1.8 with a PIKfyve inhibitor to reverse inflammatory and neuropathic pain.

使用 PIKfyve 抑制剂靶向 Na(v)1.7 和 Na(v)1.8 来逆转炎症性和神经性疼痛

Rodríguez-Palma Erick J, Loya-Lopez Santiago, Min Sophia M, Calderon-Rivera Aida, Gomez Kimberly, Khanna Rajesh, Axtman Alison D

Cellular Selectivity Analyses Reveal Distinguishing Profiles for Type II Kinase Inhibitors

细胞选择性分析揭示了II型激酶抑制剂的独特特征

Binder, Matthew J; Bashore, Frances M; Hoffman, Kaitlin K Dunn; Daamgard, Cameron; Slater, Michael R; Drewry, David H; Robers, Matthew B; Axtman, Alison D

Development of a chemical probe to enable characterization of the casein kinase 1γ subfamily

开发一种化学探针,用于表征酪蛋白激酶1γ亚家族

Capener, Jacob L; Kramer, Thomas W; Bashore, Frances M; Flory, Emily; Li, Fengling; Strang, Blair L; Axtman, Alison D

Illuminating function of the understudied druggable kinome

揭示鲜为人知的可成药激酶组的关键功能

Gomez, Shawn M; Axtman, Alison D; Willson, Timothy M; Major, Michael B; Townsend, Reid R; Sorger, Peter K; Johnson, Gary L

Discovery and optimization of narrow spectrum inhibitors of Tousled like kinase 2 (TLK2) using quantitative structure activity relationships

利用定量构效关系发现和优化窄谱Tousled样激酶2 (TLK2) 抑制剂

Asquith, Christopher R M; East, Michael P; Laitinen, Tuomo; Alamillo-Ferrer, Carla; Hartikainen, Erkka; Wells, Carrow I; Axtman, Alison D; Drewry, David H; Tizzard, Graham J; Poso, Antti; Willson, Timothy M; Johnson, Gary L

Synthesis of 5-Benzylamino and 5-Alkylamino-Substituted Pyrimido[4,5-c]quinoline Derivatives as CSNK2A Inhibitors with Antiviral Activity

合成5-苄氨基和5-烷基氨基取代的嘧啶并[4,5-c]喹啉衍生物作为具有抗病毒活性的CSNK2A抑制剂

Asressu, Kesatebrhan Haile; Smith, Jeffery L; Dickmander, Rebekah J; Moorman, Nathaniel J; Wellnitz, James; Popov, Konstantin I; Axtman, Alison D; Willson, Timothy M

Illumination of understudied ciliary kinases

对研究不足的纤毛激酶的揭示

Flax, Raymond G; Rosston, Peter; Rocha, Cecilia; Anderson, Brian; Capener, Jacob L; Durcan, Thomas M; Drewry, David H; Prinos, Panagiotis; Axtman, Alison D