日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Exponentiated model of drug demand is preferred over exponential models in people with daily/near daily cannabis use

对于每日/几乎每日使用大麻的人群,药物需求的指数模型优于指数模型。

Tolbert, Preston T; Ramirez, Miranda P; Strickland, Justin C; Lile, Joshua A; Stoops, William W; Stamper, Brady J; Sumner, Caroline B; Wesley, Michael J

An orally available non-nucleotide STING agonist with antitumor activity

一种具有抗肿瘤活性的口服非核苷酸 STING 激动剂

Bo-Sheng Pan #, Samanthi A Perera #, Jennifer A Piesvaux #, Jeremy P Presland #, Gottfried K Schroeder #, Jared N Cumming #, B Wesley Trotter #, Michael D Altman, Alexei V Buevich, Brandon Cash, Saso Cemerski, Wonsuk Chang, Yiping Chen, Peter J Dandliker, Guo Feng, Andrew Haidle, Timothy Henderson, 

Discovery of N-(Indazol-3-yl)piperidine-4-carboxylic Acids as RORγt Allosteric Inhibitors for Autoimmune Diseases

发现 N-(吲唑-3-基)哌啶-4-羧酸作为 RORγt 变构抑制剂用于治疗自身免疫性疾病

Zhang, Hongjun; Lapointe, Blair T; Anthony, Neville; Azevedo, Rita; Cals, Jos; Correll, Craig C; Daniels, Matthew; Deshmukh, Sujal; van Eenenaam, Hans; Ferguson, Heidi; Hegde, Laxminarayan G; Karstens, Willem Jan; Maclean, John; Miller, J Richard; Moy, Lily Y; Simov, Vladimir; Nagpal, Sunil; Oubrie, Arthur; Palte, Rachel L; Parthasarathy, Gopal; Sciammetta, Nunzio; van der Stelt, Mario; Woodhouse, Janice D; Trotter, B Wesley; Barr, Kenneth

Optimization of Versatile Oxindoles as Selective PI3Kδ Inhibitors

优化多功能吲哚类化合物作为选择性PI3Kδ抑制剂

Methot, Joey L; Achab, Abdelghani; Christopher, Matthew; Zhou, Hua; McGowan, Meredeth A; Trotter, B Wesley; Fradera, Xavier; Lesburg, Charles A; Goldenblatt, Peter; Hill, Armetta; Chen, Dapeng; Otte, Karin M; Augustin, Martin; Shah, Sanjiv; Katz, Jason D

Solution-Processed BiI(3) Films with 1.1 eV Quasi-Fermi Level Splitting: The Role of Water, Temperature, and Solvent during Processing

溶液法制备准费米能级分裂为1.1 eV的BiI(3)薄膜:水、温度和溶剂在制备过程中的作用

Williamson, B Wesley; Eickemeyer, Felix T; Hillhouse, Hugh W

Identification of an allosteric binding site for RORγt inhibition

鉴定RORγt抑制剂的变构结合位点

Marcel Scheepstra ,Seppe Leysen ,Geert C van Almen ,J Richard Miller ,Jennifer Piesvaux ,Victoria Kutilek ,Hans van Eenennaam ,Hongjun Zhang ,Kenneth Barr ,Sunil Nagpal ,Stephen M Soisson ,Maria Kornienko ,Kristen Wiley ,Nathaniel Elsen ,Sujata Sharma ,Craig C Correll ,B Wesley Trotter ,Mario van der Stelt ,Arthur Oubrie ,Christian Ottmann ,Gopal Parthasarathy ,Luc Brunsveld

Characterization of non-nitrocatechol pan and isoform specific catechol-O-methyltransferase inhibitors and substrates

非硝基儿茶酚泛和异构体特异性儿茶酚-O-甲基转移酶抑制剂和底物的表征

Ronald G Robinson, Sean M Smith, Scott E Wolkenberg, Monika Kandebo, Lihang Yao, Christopher R Gibson, Scott T Harrison, Stacey Polsky-Fisher, James C Barrow, Peter J Manley, James J Mulhearn, Kausik K Nanda, Jeffrey W Schubert, B Wesley Trotter, Zhijian Zhao, John M Sanders, Robert F Smith, Debra M

Replicating satellite RNA induces sequence-specific DNA methylation and truncated transcripts in plants

复制型卫星RNA在植物中诱导序列特异性DNA甲基化和截短转录本的产生。

Wang, M B; Wesley, S V; Finnegan, E J; Smith, N A; Waterhouse, P M