Discovery of N-(Indazol-3-yl)piperidine-4-carboxylic Acids as RORγt Allosteric Inhibitors for Autoimmune Diseases
发现 N-(吲唑-3-基)哌啶-4-羧酸作为 RORγt 变构抑制剂用于治疗自身免疫性疾病
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.9b00431
Zhang, Hongjun; Lapointe, Blair T; Anthony, Neville; Azevedo, Rita; Cals, Jos; Correll, Craig C; Daniels, Matthew; Deshmukh, Sujal; van Eenenaam, Hans; Ferguson, Heidi; Hegde, Laxminarayan G; Karstens, Willem Jan; Maclean, John; Miller, J Richard; Moy, Lily Y; Simov, Vladimir; Nagpal, Sunil; Oubrie, Arthur; Palte, Rachel L; Parthasarathy, Gopal; Sciammetta, Nunzio; van der Stelt, Mario; Woodhouse, Janice D; Trotter, B Wesley; Barr, Kenneth